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3-({methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}methyl)pyrrolidin-3-ol
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-(1,3-thiazol-5-ylmethyl)pyrrolidine-2-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-methyl-5-[4-(methylsulfanyl)phenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
N-ethyl-6-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-3-carboxamide
(2S,4R)-1-methyl-4-(5-phenylpentanamido)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-phenylpiperidine-4-carbonitrile
N-{2-cyclobutyl-7-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide
5-ethyl-N,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
2-(3,4-difluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-methyl-4-{[5-(5-methyl-1,2-oxazol-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
2-{[(3R,5S)-5-(4-methyl-1,4-diazepane-1-carbonyl)-1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
(1S,5R)-6-cyclobutanecarbonyl-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-methyl-2-(5-phenylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{1-[(4-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}-1λ6-thiolane-1,1-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(2-fluorophenyl)pyrrolidin-1-yl]butan-1-one
N-methyl-2-(pyridin-3-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
methyl 4-methyl-3-({[3-(oxolan-3-yl)propyl]carbamoyl}amino)benzoate
4-(cyclopropylamino)-5-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(methanesulfonylmethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine
7-chloro-3-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
4-methoxy-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2,5-dimethyl-N-{2-[5-methyl-4-({2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-3-carboxamide
N-{1-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}pyridine-3-carboxamide
(3S,4S)-1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(4-fluorophenyl)piperidin-3-ol
N-{[5-(methoxymethyl)furan-2-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
4-(1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine-4-carboxylic acid
3-(2-methoxyphenyl)-N-[2-(1H-pyrazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-(cyclohexylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N3-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-1,3-dicarboxamide
2-[(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidin-4-yl)formamido]acetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,6-dimethylquinoline-3-carboxamide
(3R,4R)-1-(6-chloro-2H-chromene-3-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
1-[(4-methoxyphenyl)methyl]-4-[3-(methylsulfanyl)butyl]piperazin-2-one
5-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-2-methoxyphenol
6-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(9H-fluoren-9-yl)-2-oxo-6-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
3-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)phenol
3-[1-(1,3-thiazol-2-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
N-{4-[(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenyl}acetamide
3,3,3-trifluoro-2-hydroxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methylpropanamide
2-(4-ethoxyphenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole