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5-acetyl-N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
2-(2-butyl-1H-imidazol-4-yl)-1-methyl-1H-1,3-benzodiazole
N-(3,5-dimethoxyphenyl)-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
{2-[4-(3-fluoro-2-methylphenyl)-1H-1,2,3-triazol-1-yl]-1-(5-methylfuran-2-yl)ethyl}dimethylamine
3-(2-fluorophenyl)-1-(1,2-oxazinan-2-yl)-3-phenylpropan-1-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2,6-dimethyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylacetamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidine
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 2-{N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamido}acetate
2-(2-ethyl-1H-imidazol-1-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(4-hydroxyphenyl)ethyl]-1,3-oxazole-4-carboxamide
2-({2-amino-6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}acetamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}propanamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-amino-4-(5-chloro-3-methoxy-2-propoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-[(2,6-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-(3-{[ethyl(methyl)amino]methyl}phenoxy)propan-2-ol
3-{2-oxo-2-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-(3-methoxypropyl)-1-methyl-N-[3-(4-methylphenyl)propyl]piperidin-4-amine
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-[(3-acetylphenyl)methyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
1-(cyclopropylmethyl)-4-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-2-(propan-2-yl)-1,4-diazepane
2-phenyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
5-(1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
N-[(3,4-difluorophenyl)methyl]-3-[1-(3-methoxypropanoyl)piperidin-3-yl]propanamide
4-(2-{1-[(4-methanesulfonylphenyl)methyl]piperidin-2-yl}ethyl)phenol
1-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-2-(morpholin-4-yl)ethan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-1-(3-hydroxyazetidin-1-yl)ethan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-ethylpyrrolidine-2-carboxamide
2-[5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(6-ethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-phenyl-4-[2-(3-phenylpyrrolidin-1-yl)acetyl]piperazin-2-one
6-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2-ethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(propan-2-yl)-1H-pyrazole-4-amido]pyrrolidine-3-carboxylic acid
3-[(3aS,6aS)-1-[(6-methylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(1R,3S)-3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]cyclopentan-1-amine
2-cyclopropyl-4-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrimidine-5-carboxamide
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
6-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[1-ethyl-2-(2-fluorophenyl)-5-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
1-(oxan-4-ylmethyl)-2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
2-(4-methyl-1H-pyrazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one