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3,5,7-trimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-indole-2-carboxamide
5-tert-butyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,3,4-oxadiazol-2-amine
(2R,6S)-2,6-dimethyl-4-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]morpholine
5-acetyl-N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methylthiophene-3-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-(2-methylpyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
4-(1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}azetidin-3-yl)morpholine
N-[(1R,2R)-2-hydroxycyclohexyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-propylpropanamide
1-[2-(propan-2-yl)pyrimidine-5-carbonyl]azocane
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[3-(methylsulfanyl)phenyl]urea
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]pyrrolidine-1-carboxamide
(3aR,6aR)-2-acetyl-5-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(8-hydroxyquinolin-2-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclohexyl-6-(pyridin-4-ylmethoxy)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
N-(1-cycloheptylpiperidin-3-yl)propanamide
N-cyclopropyl-3-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]sulfonyl}benzamide
3-(azepane-1-carbonyl)-5-(4-ethylpiperazin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(hydroxymethyl)piperidin-3-yl)methanol
1-(4-fluorobenzoyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-ethyl-2-(2-fluorophenoxymethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
1,5-dimethyl-4-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[2-hydroxy-2-(naphthalen-2-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[3-(azetidin-1-ylmethyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(3,4,5-trifluorophenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[1-(2,4-dimethylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
2-[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]acetamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
5-acetyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}thiophene-2-carboxamide
1-[2-(pyridin-2-yl)-4-{[3-(pyridin-4-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-[4-(methylsulfanyl)benzoyl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
N-[(1R,3R)-3-aminocyclopentyl]-2-methyl-2-[(4-methylphenyl)amino]propanamide
N3-(2-methylpropyl)-N3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-1,3-dicarboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{3-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]phenyl}ethan-1-one
2-(ethanesulfonyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-cyclopropyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-cyclopentyl-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
7-(2-methoxyphenyl)-2-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-hydroxyethyl)-5-(2-methyloxane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-N-ethyl-N-methylpyrimidin-4-amine
2-(4-chlorophenoxy)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-[(4-chlorophenyl)methyl]-3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propanamide
2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propane-1,3-diol
(1S,5R)-1,3,3-trimethyl-N-[2-(morpholin-4-ylmethyl)phenyl]-6-azabicyclo[3.2.1]octane-6-carboxamide
4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]-1λ6-thiomorpholine-1,1-dione
N-{4-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}acetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide