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[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]pyrrolidin-3-yl]methanol
2-ethyl-1-[1-methyl-4-(2-phenylethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]butan-1-one
2-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]thiophene-3-sulfonamide
5-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]pyridine-2-carbonitrile
(1R,9S)-5-amino-12-methyl-3-(6-methyl-2H-1,3-benzodioxol-5-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
4,5-dimethyl 1-[(3S,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-{[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2,2-dimethyloxan-4-amine
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
1-ethyl-5-{[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-(2-hydroxyphenyl)-N-methylacetamide
4-{4-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-1-yl}benzonitrile
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(furan-2-carbonyl)-1,4-diazepane
4-(1-ethyl-1H-imidazol-2-yl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
1-cyclopropanecarbonyl-N-[3-(4-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-methoxyethyl)-3-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)propanamide
N-({1-[1-(prop-2-yn-1-yl)piperidin-4-yl]piperidin-3-yl}methyl)-1,2,5-oxadiazole-3-carboxamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
3-(2-chlorophenyl)-1-methyl-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
methyl[(3-methyl-1H-pyrazol-4-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine
2-(3-methylphenyl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
2-(2-hydroxyethyl)-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroquinolin-2-one
N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}cyclopropanamine
N-[(5-chloro-1H-indol-2-yl)methyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
7-cyclohexyl-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
1-(4-chloro-2,5-dimethylbenzenesulfonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-(5-acetylthiophen-3-yl)-N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[2-(1H-imidazol-1-yl)-1-phenylethyl]urea
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(dimethylamino)-2-{4-[(2-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
2-{2-[(dimethylamino)methyl]phenoxy}-N-ethylpyridine-4-carboxamide
(2S,4R)-4-amino-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperidin-3-yl]-3-phenylpropan-1-one
(S)-[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl](phenyl)methanol
(3aR,6aR)-2-cyclohexyl-5-(6-methylpyridine-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
9-methoxy-7-oxo-3-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-methyl-1-(2-methylpropyl)-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
methyl (2S,4R)-1-methyl-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-amido]pyrrolidine-2-carboxylate
(3S,4S)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
[(3R,4R)-1-(dimethyl-1,3-thiazol-2-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-methoxyphenoxy)acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-2-ylsulfanyl)acetamide