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(2S,4S)-1-benzyl-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-4-phenylbenzamide
4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
[(3,5-dimethoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(5-methylthiophene-2-carbonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-fluorophenyl)-5-[4-(propan-2-yloxy)benzoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-ethyl-2-methyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine
2-benzyl-N-(1,4-dioxan-2-ylmethyl)-1,3-thiazole-4-carboxamide
5-(2-fluorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-[3-(prop-2-en-1-yloxy)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(furan-2-yl)propanamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-N-propyl-1,2-dihydroquinoline-4-carboxamide
(3R,4R)-1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(3S,4S)-4-cyclopropyl-1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
2,4-dimethoxy-6-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrimidine
8-(2-amino-6-methylpyrimidin-4-yl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-cyclopentylpiperidine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N,N-diethyl-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-imidazol-2-ylmethyl)piperidine
2-benzyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1,3-thiazole-4-carboxamide
2-chloro-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-acetamido-N-methylbenzamide
methyl 4-{5-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-2-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-cyclopentylethan-1-one
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-3-yl]methanol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]benzamide
1-(1-carbamoylcyclopropanecarbonyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(3R,4R)-3-hydroxy-1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-4-yl]pyridine-4-carboxamide
2-(2-methoxy-5-methylphenyl)-2-[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]acetic acid
N-[(2-fluorophenyl)methyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
N-(1,4-dioxan-2-ylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
N-(3-methyl-1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
1-(azepan-1-yl)-3-[3-({methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[2,5-dioxo-4-(pyridin-3-yl)imidazolidin-4-yl]piperidin-1-yl}acetic acid
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2,6-dimethoxyphenol
(1S,2S,9S)-N-[3-(1H-imidazol-5-yl)phenyl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}adamantane-1-carboxamide
N-(2,5-dimethoxyphenyl)-3-[4-(2-methylpropyl)piperazin-1-yl]-3-oxopropanamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-hydroxy-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
2-{2-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenoxy}ethan-1-ol
3-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}benzamide
methyl 2-{2-[(2-methoxyacetamido)methyl]-5-methyl-2,3-dihydro-1-benzofuran-7-yl}benzoate
methyl 1-[3-(4-{[bis(prop-2-en-1-yl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidine-4-carboxylate