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2-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-3-carbonitrile
3-[2-(azocan-1-yl)-2-oxoethyl]-1-benzyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-(2-hydroxyethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(oxan-4-yl)ethyl]propanamide
(2R)-2-amino-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(ethylsulfanyl)propan-1-one
1-(1-benzofuran-5-ylmethyl)-4-(3-methoxybenzoyl)piperazine
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-(oxolan-3-ylmethyl)acetamide
2-{4-[(2-chlorophenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-benzothiazole-6-sulfonamide
4-(5-methylpyridin-2-yl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-ol
5-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]-N-phenylpyridin-2-amine
4-ethyl-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(hydroxymethyl)-2-methyl-4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)pyridin-3-ol
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propane-1-sulfonamide
2-{[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl}-1-(propan-2-yl)-1H-1,3-benzodiazole
N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
3-{[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]methyl}benzonitrile
6-{methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-(3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)pyrimidine
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxy-2-phenylacetamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
N-methyl-1-(piperidin-3-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzoxazole
N-ethyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzamide
5-(2,6-difluorophenoxymethyl)-3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
3-{3-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
1-amino-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}cyclopropane-1-carboxamide
3-methyl-9-[3-(1H-1,2,4-triazol-5-yl)benzoyl]-3,9-diazaspiro[5.6]dodecane
8-(6-aminopyrimidin-4-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4S)-1-[2-(1H-imidazol-2-yl)benzoyl]-4-propylpyrrolidine-3-carboxylic acid
1-{4-[(2,6-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
2-ethyl-5-[3-(piperidin-1-yl)azetidine-1-carbonyl]pyrimidine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-cyclopentyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-phenoxypyridin-3-yl)methyl]oxolane-3-carboxamide
N-{[1-(carbamoylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}-2-methoxybenzamide
2-methoxy-N,4-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
2-{[4-(2-fluorophenyl)-5-(1H-indol-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(4-methoxyphenyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
N-[(2R,3R)-1'-[(2,5-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
4-hydroxy-2-[(4-methanesulfonylpiperazin-1-yl)methyl]quinoline-6-carboxamide
5-({2-cyclobutanecarbonyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)-N-propylpyrimidin-2-amine
5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine