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6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-[(2S)-2-hydroxypropyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(5-ethylthiophene-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-methylpiperazin-1-yl)propanamide
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
N-(propan-2-yl)-5-[1-(pyridazine-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-{2-hydroxy-3-[4-methoxy-2-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
3-{4-[(5-chlorofuran-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
2-{3-[({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}carbamoyl)amino]phenyl}acetamide
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-4-sulfamoylbenzamide
2-amino-4-(4-hydroxy-2-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
6-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydroquinolin-4-one
5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propanamide
5-chloro-2-methyl-3-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-indole
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)oxan-4-amine
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2,4-difluorophenyl)methyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
5-methyl-2-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
4-[3-(2-oxopyrrolidin-1-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
1-methyl-2-oxo-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1H-1,2,4-triazole
N1-tert-butyl-N2-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1,2-dicarboxamide
3-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
1-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-3-methylbut-2-en-1-one
3-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methoxyethoxy)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]-6-methyl-1,2-dihydropyridin-2-one
2-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]thiophene-3-sulfonamide
2-methyl-8-(pyrrolidine-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-chloro-2-(furan-2-yl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-4-carboxamide
N5-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidine
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
2-ethyl-4-phenyl-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecane
(3R,5S)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(3R,4R)-1-(5-chloropyridin-2-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
1-[4-(benzyloxy)piperidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-[2-(4-methoxyphenyl)ethyl]-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
5-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-{2-[(1-hydroxy-2-methylpropan-2-yl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
methyl 4-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)benzoate
N-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}methanesulfonamide
4-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-1,2,5-oxadiazole-3-carboxamide
(5S,9aS,9bS)-5-(5-acetylthiophen-3-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[3-(3-fluorophenyl)phenyl]-1-(pyrrolidine-2-carbonyl)piperidine-4-carboxamide