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(3S,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
N-(propan-2-yl)-5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
4-ethyl-1-methyl-3-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-methanesulfonylacetamido)-4-methylphenyl]pentanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,5-dimethylthiophene-2-carboxamide
2-(dimethylamino)-N-methyl-N-(2-phenyl-1-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl)acetamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(2-oxoimidazolidin-1-yl)benzamide
3-methyl-N-(1-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
5,5-dimethyl-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-oxazolidine-2,4-dione
3-(1-benzyl-1H-pyrazole-4-carbonyl)-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
1-methyl-N-(3-methylphenyl)-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-[(3-chlorophenyl)methyl]-N-(2-hydroxypropyl)-1,3-benzoxazole-6-carboxamide
(2S,4R)-N-(2-methoxyethyl)-1-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
methyl 2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)-4-(methylsulfanyl)butanoate
(2-{[4-(cyclopentylmethyl)piperazin-1-yl]methyl}phenyl)methanol
N-{[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl 4-[4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]benzoate
N-(9H-fluoren-9-yl)-6-({4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(5-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
3-(2-phenylethyl)-N-(thiophen-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[3-(3-methoxypiperidin-1-yl)-3-oxopropyl]-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
5-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)pyridine
{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-benzyl-1-cyclohexyl-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
6-(4-methoxy-2-methylphenyl)quinazolin-4-amine
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[2-(thiophen-3-yl)acetamido]methyl}benzoate
(1S,3R)-3-(3-methoxypropanamido)-N-[2-(4-methylphenyl)ethyl]cyclopentane-1-carboxamide
4-{[2-(furan-3-yl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1-(propan-2-yl)-1H-pyrazole
2-(4-methoxyphenoxy)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]pyridazine-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(3R,4R)-1-(1H-imidazol-2-ylmethyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-(4-fluorophenoxymethyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
3-(3-phenylpropyl)-1-(1,3-thiazol-2-yl)piperidine-3-carboxylic acid
2-(pyridin-3-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
5-(6-hydroxy-4-propyl-1,4-diazepane-1-carbonyl)-1H-pyrrole-3-carbonitrile
3-(3-methoxyphenyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
(1s,4s)-4-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]cyclohexan-1-ol
1-(1-benzofuran-2-ylmethyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
{1-[2-({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-2-yl}methanol
3-{2-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(3-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 6-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}-3-(2-methylpropanamido)thieno[2,3-b]pyridine-2-carboxylate
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide