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2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}propanamide
methyl 6-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}pyrazine-2-carboxylate
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)methanol
N-[3-(4-fluorophenyl)phenyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(pyridin-4-ylsulfanyl)acetamide
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1-(3-hydroxyphenyl)pyrrolidin-2-one
N-[3-(furan-2-yl)phenyl]-1-(2-oxo-2-phenylacetyl)piperidine-4-carboxamide
2-(furan-2-yl)-1-[(2,4,6-trimethoxyphenyl)methyl]azepane
5-(8-methoxyquinolin-2-yl)pyridin-2-amine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-3-(thiophen-2-yl)propanamide
1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-(3,5-dimethoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
methyl 1-[2-(1H-indol-3-yl)ethyl]-5-{[(4-methoxyphenyl)methyl]amino}-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(5S,9aS,9bS)-5-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N'1-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopropane-1,1-dicarboxamide
2-[5-cyclopropyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2,5-dimethylthiophen-3-yl)pyrimidine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,2-dihydrophthalazin-1-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,4-diazepan-5-one
(3S,9aR)-3-benzyl-2-methyl-8-(thiophen-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
2-[5-(2-chlorophenyl)-1H-indazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}-6-chloroimidazo[2,1-b][1,3]thiazole
4-{ethyl[2-(4-methoxyphenoxy)ethyl]amino}butan-1-ol
1-(3-{[(cyclopropylmethyl)(propyl)amino]methyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
1-{3-[3-(1-methoxyethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
N-(1-phenylcyclopropyl)thieno[2,3-d]pyrimidin-4-amine
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine-4-carboxylate
1-{[2-(dimethylamino)-2-(3-methylphenyl)acetamido]methyl}cyclopentane-1-carboxylic acid
3-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)-1,3-oxazolidin-2-one
5-methyl-1-(2-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclopropylmethyl)-5-(5-methoxyfuran-2-carbonyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4,6-dimethyl-3-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
4-chloro-1-methyl-3-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indazole
2-(2H-1,2,3-benzotriazol-2-yl)-1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)ethan-1-one
5-benzyl-5-(1-propylpiperidin-4-yl)-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
4-ethyl-1-methyl-3-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-(1H-pyrazol-1-yl)-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]butan-1-one
N-[(1-cyclopentylpyrrolidin-3-yl)methyl]-2-(3,5-dioxomorpholin-4-yl)acetamide
N-[2-(pyridin-3-yloxy)ethyl]naphthalene-2-carboxamide
N-ethyl-6-fluoro-2-(2-methylpyrimidin-5-yl)-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
N-[(2R,3R)-1'-(dimethyl-1,3-thiazole-5-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
[(3R,4R)-1-(2,6-difluoro-3-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
(1R,5R)-3-methanesulfonyl-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane