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4-(1H-imidazol-1-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]butan-1-one
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)oxane-4-carboxamide
5-(2,6-difluorophenoxymethyl)-N-(1-phenylcyclopropyl)-1,2-oxazole-3-carboxamide
9-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-[(diethylcarbamoyl)methyl]-N-(2-phenoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-[({3-[2-(dimethylcarbamoyl)ethyl]phenyl}carbamoyl)amino]cycloheptane-1-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)methyl]-1H-indole-2-carboxamide
3-(3,4-dimethoxyphenyl)-N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
1-ethyl-5-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-2-one
3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1-(1H-1,2,4-triazol-3-yl)urea
N-(2-benzylbutyl)-1-methylpiperidin-4-amine
1-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3-dihydro-1H-indene-1-carboxamide
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-({8-[(4-methoxynaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(1R,7S)-3-cycloheptyl-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-cyclohexyl-4-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
ethyl 3-(3-phenylpropyl)-1-[3-(pyridin-2-yl)propanoyl]piperidine-3-carboxylate
(2R,3S,6R)-3-(4-fluorophenyl)-5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(piperidine-1-carbonyl)phenoxy]-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
7-(3-chlorophenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-{2-[cyclopentyl(methyl)amino]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[2-(dimethylamino)ethyl]-9-(3-hydroxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-(1H-indole-6-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-[3-(furan-2-yl)propyl]-1-methylazepane-2-carboxamide
3-(1H-pyrazol-5-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
1-(3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
1-[7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
5-(4-methoxyphenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(1-methylpiperidin-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-phenyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
N-[4-(furan-2-yl)butan-2-yl]-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-amine
6-[({[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
2-[3-(2-amino-3-cyano-6-cyclopentyl-5-methylpyridin-4-yl)phenoxy]acetamide
2-(4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
2-[2-(dimethylamino)ethyl]-8-[2-(3-methylphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one