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2-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-6-methylpyridine
N-[(4-chlorophenyl)methyl]-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(1H-1,2,4-triazol-3-yl)benzamide
9-ethyl-1-methyl-4-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-methyl-1,3-thiazol-2-yl)-4-(piperidine-1-carbonyl)piperidine
5-{1-[(2-ethoxypyridin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-[(6-methylquinolin-5-yl)methyl]piperidin-3-yl]propanoic acid
4-methanesulfonyl-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]benzamide
N-[(2S,4R,6S)-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-({8-[(2,5-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxyacetamide
1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-methylpiperazine
1-cyclohexyl-3-(4-fluorophenoxymethyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-phenyl-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-N3-methyl-4-oxo-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
2-(4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperazin-1-yl)-N-phenylacetamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[4-(methylamino)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidine-3-carboxylic acid
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2,1,3-benzoxadiazole
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
5-(2-{[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
(3S,4S)-4-cyclopropyl-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
1-(2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
4-cyclopropanecarbonyl-N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
3-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-3,5-dimethyl-1H-pyrazol-4-yl)benzoic acid
N-methyl-N-(2-{[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}ethyl)methanesulfonamide
7-(2-hydroxyethyl)-2-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(2-methoxyethyl)(methyl)amino]-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-(furan-2-yl)propan-1-one
3-{1-oxaspiro[4.5]decan-3-yl}-1-[4-(1H-pyrazol-4-yl)phenyl]urea
1-[(2,4-dimethyl-5-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}phenyl)methyl]-4-methylpiperidine
1-(2-methoxyphenyl)-4-[1-(4-methylbenzenesulfonyl)piperidin-3-yl]piperazine
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(cyclohexylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-2,5-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-ethylpiperidine-1-carboxamide
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
(3aS,6aS)-2-(oxan-4-yl)-5-(1,3-thiazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(3-methoxypropyl)amino]-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(adamantan-2-yl)-N-phenylpiperidin-3-amine
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
1-(3-fluorophenyl)-3-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
3-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-oxopropyl)-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
12-[4-(2-methoxyethyl)piperazine-1-carbonyl]-15-methyl-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
1-[2-methoxy-5-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol