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4-{[(5-methyl-1,3,4-oxadiazol-2-yl)amino]methyl}benzene-1-sulfonamide
2-{4-[5-(2-chlorophenyl)furan-2-yl]-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}phenol
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
6-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
ethyl[(1-methyl-1H-imidazol-2-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(2S,4S)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N,1-dimethyl-3-(2-methylpropyl)-N-(thian-4-yl)-1H-pyrazole-5-carboxamide
3-(2,4-dimethoxyphenyl)-4-methylpyridine
N-[(3R,4R)-3-hydroxy-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]pyrazine-2-carboxamide
[(3-ethoxy-4-methoxyphenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yl)ethyl]amine
3-(2,3-dimethoxyphenyl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine
1-cyclopropyl-4-{[2-(8-methoxyquinolin-2-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-(pentan-3-yl)piperidine
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-phenylbutane-1,4-dione
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(2,5-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
1-(3-{[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propyl)pyrrolidin-2-one
N-[2-(1H-imidazol-1-yl)ethyl]-2-(oxan-2-ylmethoxy)acetamide
2-hydroxy-N-[2-(1-methylpiperidin-3-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-methyl-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(1H-indol-2-ylmethyl)piperidine-4-carboxamide
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole
[(3R,4R)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[2-(pyridin-3-yloxy)propyl]acetamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[(4-fluorophenyl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)ethan-1-amine
(1S,5R)-6-benzyl-3-(3-fluoropyridin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
methyl 2-[bis(prop-2-en-1-yl)sulfamoyl]-6-(quinolin-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(6-cyanopyridin-3-yl)-4-cyclobutanecarbonyl-1,4-diazepane-1-carboxamide
6-(propan-2-yl)-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
2-chloro-6-fluoro-N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
2-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}propanamide
4-(pyridin-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-2-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(1H-imidazol-2-yl)benzamide
5-(2,4-difluorophenoxymethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(4-methylpiperazin-1-yl)propan-1-one
N-[2-(dimethylamino)ethyl]-4,4,4-trifluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)butanamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-(4,6-dimethylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
methyl 2-(4-{[bis(prop-2-en-1-yl)carbamoyl]methyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
5-methyl-3-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1H-indazole