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2-{[5-(3-methylthiophen-2-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[2-(2-methylphenoxy)ethyl]urea
[4-(2-cyclopropylquinoline-4-carbonyl)-1,4-oxazepan-6-yl]methanol
(1S,4S)-5-[(2S)-2-aminopropanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-methylphenyl)quinoline-4-carboxamide
N-(1-acetylpiperidin-4-yl)-3-(3-hydroxy-3-methylbutyl)benzamide
2-(dimethylamino)-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]pyrrolidin-3-ol
1-{4-[(4-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
2-{4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-methylpiperazin-2-yl}ethan-1-ol
(2S)-2-amino-3-methoxy-N-[2-(3-phenylpropoxy)phenyl]propanamide
2-methyl-8-(5-propylthiophene-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{4-[2-(2,4-dimethylphenoxy)ethyl]phenyl}-N-methylacetamide
2-{[3-(N-methylacetamido)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-methyl-N-[(5-methylfuran-2-yl)methyl]-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-(3,5-dimethylphenyl)-N'-{2-[(pyridin-3-yl)amino]ethyl}propanediamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-8-methylimidazo[1,2-a]pyridine-2-carboxamide
N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide
4-[(3-fluorophenyl)methyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
methyl 8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(3S)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-N,N-dimethylazepan-3-amine
methyl 3-(2-methoxybenzamido)-5-{[2-(2-methylphenyl)acetamido]methyl}benzoate
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,2,6-trimethylquinoline-4-carboxamide
3-{[4-(dimethylamino)azepan-1-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
2-{1-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1,3-benzoxazole
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-{[4-(benzyloxy)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(3-chlorophenyl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
1-[(2-aminopyridin-3-yl)methyl]-4-(9H-purin-6-yl)-1,4-diazepan-6-ol
8-methyl-2-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]-2,8-diazaspiro[4.5]decane
1-ethyl-1-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
4-{[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-1λ6-thiane-1,1-dione
N-methyl-3-({4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)pyridin-2-amine
({4-ethyl-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-ethylpiperidine
2-[benzyl(methyl)amino]-N-[2-(pyrrolidin-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-(furan-2-yl)-5-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}pyrimidine
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-ethyl-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-(propan-2-yl)-1H-pyrazole
4-[1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperazine-1-carbaldehyde
2-(2-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
(2S)-2-{[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-phenylpropanamide
3-[(3R,4S)-1-(1-benzofuran-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
9-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-4,6-dimethyl-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)furan-3-carboxamide