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N-{2-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-4-methylphenyl}benzamide
N-[(2R,3R)-1'-(4-methoxybenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
methyl 4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)piperidine-1-carboxylate
1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
4-ethyl-6-[3-(pyridin-4-yl)azetidin-1-yl]-2-(pyrrolidin-1-yl)pyrimidine
6-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-6-methylpyridine
2-cyclopropyl-9-(3,4-dimethylbenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-benzyl-5-methanesulfonamido-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
4-(azepane-1-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
4-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-[(1H-1,3-benzodiazol-2-ylmethyl)(benzyl)amino]-2-methylpropan-1-ol
1-(3-{3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazol-4-yl}phenyl)ethan-1-one
N-methyl-N-[(4-methylphenyl)methyl]-3-(3-methylpiperidin-1-yl)propanamide
N-(1H-indol-2-ylmethyl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
5-[butyl(methyl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(4-fluorophenyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
7-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-1,2-dihydroisoquinolin-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
4-(2-fluorophenoxy)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
2-[4-(1,3-benzothiazol-2-yl)-1,4-diazepane-1-carbonyl]-6-methyl-4H-pyran-4-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(pyrrolidine-1-carbonyl)piperidine
3-(3-methylbut-2-en-1-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine-3-carboxylic acid
4-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(3-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-[(3S,4R)-1-benzyl-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
2-[4-(butane-1-sulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
N-(2-hydroxyethyl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-(quinolin-5-ylmethyl)propanamide
(1S,5R)-6-(2-methoxyethyl)-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N'1-(4-pentanamidophenyl)cyclopropane-1,1-dicarboxamide
3-(2,3-dihydro-1H-inden-4-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-6-oxo-1,6-dihydropyridine-2-carboxamide
3-methyl-8-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1H-inden-2-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{2-[methyl(phenyl)amino]ethyl}cyclopentane-1,3-dicarboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
5-[(dimethylamino)methyl]-N-[(4-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)furan-2-carboxamide
(2S,4S)-4-amino-1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide