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benzyl({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}propanamide
N-cyclopentyl-6-(dimethylamino)-N-[(5-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
4-(1H-imidazol-2-ylmethyl)-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-benzothiophen-5-ylmethyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyridin-4-yl)propyl]benzamide
5-{[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
4-(4-{[3-(phenylamino)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-ethyl-N,2-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]quinoline-4-carboxamide
1-(1-methylpiperidine-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-3-yl)ethyl]propanamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-ethyl-N-methyl-N-(quinolin-5-ylmethyl)thiophene-3-carboxamide
N-methyl-N-(oxan-4-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-({2-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N4-(pyridin-4-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N,N-dimethyl-3-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]sulfamoyl}benzamide
1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
1-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
(4aS,8aR)-6-(4-aminobutanoyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(2-chlorophenoxy)azetidin-1-yl]propan-1-one
2-cyclopropyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
1-(2-methoxyethyl)-8-[(6-methylpyridin-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}dimethylamine
3-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
N-(cyclopropylmethyl)-4-[2-oxo-2-(piperidin-1-yl)ethoxy]-N-propylbenzamide
2-methyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidin-4-amine
ethyl 1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
(1S,5R)-3-(5-acetylthiophene-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-oxa-9-azaspiro[5.5]undecane
3-ethyl-5-hydroxy-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]adamantane-1-carboxamide
3-propyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[4-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one
2-[methyl(pyridin-4-ylmethyl)amino]-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
(2S,4S)-N-ethyl-1-methyl-4-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamido]pyrrolidine-2-carboxamide
N-cyclobutyl-4-(piperidin-3-yl)benzamide
4'-(3-methylbutyl)-1-[2-(1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
N-(furan-2-ylmethyl)-2-(2-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]acetamide
methyl 3-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(3-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)piperidin-2-one
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-cycloheptyl-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
5-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
3-(furan-2-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]propanoic acid
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-(benzyloxy)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidine