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2-(3,4-dimethoxyphenyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[3-(3-fluorophenyl)phenyl]-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-3-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-methoxyphenyl]ethan-1-amine
N-(3-chloro-4-ethoxyphenyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
1-(2,2-dimethyloxane-4-carbonyl)-4-(2-fluorophenyl)piperazine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpyridine-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2,4,6-trifluorophenyl)acetamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
1-(thiophen-3-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-ol
(1R,6S)-9-methyl-3-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
({4-cyclopropyl-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(5-methoxyfuran-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-(azetidine-1-carbonyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]benzene-1-sulfonamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
2-({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-N,N-dimethylethane-1-sulfonamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)piperidin-1-yl]piperidine
4-(4-methyl-1H-pyrazol-3-yl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]piperidine-1-carboxamide
{[5-(1-cyclohexanecarbonylpiperidin-4-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(cyclopropylmethyl)({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(2-methylphenyl)-1,4-diazepane
N-[(3R,5S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
3-{4-[6-(aminomethyl)-2-methylpyrimidin-4-yl]piperazin-1-yl}pyrazine-2-carbonitrile
1-[2-(3-methoxyphenyl)ethyl]-3-(5-propyl-4H-1,2,4-triazol-3-yl)urea
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-phenylethane-1,2-dione
3-[(3R,4S)-1-[(4-methanesulfonylphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-[(3R,4S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
methyl 3-({[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}(pyridin-2-ylmethyl)sulfamoyl)thiophene-2-carboxylate
1-(thiophene-2-carbonyl)-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methoxyphenyl)acetamide
3-{[4-(3-chlorophenyl)-5-({methyl[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
(2E)-3-(2-chlorophenyl)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(2,3,6-trimethylphenoxy)acetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-1-(4-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}piperidin-1-yl)propan-1-one
3-(2-methyl-1H-indol-1-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
N3-(5-methylpyridin-2-yl)-N1-[1-(propan-2-yl)piperidin-4-yl]propane-1,3-diamine
3-chloro-N-(2-methoxyethyl)-4-({1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(4-cyano-2-ethylphenyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
N,N-diethyl-1-{[(pyrazin-2-yl)carbamoyl]methyl}piperidine-3-carboxamide
2-methoxy-1-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepan-1-yl}ethan-1-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(2-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1H-pyrrole-2-carbonitrile
2-[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-N-ethylacetamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-4-oxo-N-[(3S)-2-oxoazepan-3-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(carbamoylmethyl)-N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]piperidine-4-carboxamide