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7-[2-chloro-5-(trifluoromethyl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(3-fluorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(piperidin-1-yl)butanamide
2-{2-[2-(furan-2-yl)azepan-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
4-[4-({4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-(2-methylphenyl)-4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
N-methyl-5-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-6-methylpyrimidin-2-amine
N-[(3R,4S)-1-(5,6-dimethylpyrazin-2-yl)-4-propylpyrrolidin-3-yl]-3-methoxypropanamide
methyl 4-{5-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-1,2,4-oxadiazol-3-yl}benzoate
2-[(2-methoxyphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1H-indol-1-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(3-chloro-2-fluorophenyl)methyl]-5-cyclopropyl-1,3-oxazole-4-carboxamide
4-(cyclopropylmethyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
4-chloro-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2,5-dimethoxy-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
(1R,2S)-1-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1H-inden-2-ol
5-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-6-methyl-2-(9H-purin-6-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{[4-(aminomethyl)phenyl]methyl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
2-methoxy-N-(1-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1S,5R)-3-benzoyl-6-(5-chlorothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)ethane-1-sulfonamide
4-(4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperazine-1-carbaldehyde
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
(1-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
3-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenol
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-[1-(2,5-dimethylbenzoyl)piperidin-2-yl]ethyl}morpholine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(methylsulfanyl)pyrimidine-5-carboxamide
N-(1-cyclopropylethyl)-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
(3S,4R)-4-methyl-1-[3-(5-methylfuran-2-yl)benzoyl]piperidine-3,4-diol
1-(dimethylamino)-3-[4-methoxy-2-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-({3-[(dimethylamino)methyl]phenyl}methyl)-4-sulfamoylbenzamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(2S,4S)-N-ethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-4-carboxylate
3-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
1-(2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethyl)pyrrolidin-2-one
N-methyl-N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}oxolan-3-amine
N-(3-methylphenyl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
3-fluoro-N-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-methanesulfonyl-3-methyl-3-phenylpiperidine
[2,4,6-trimethyl-3-({[2-(pyridin-4-ylformamido)ethyl]amino}methyl)phenyl]methyl acetate