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1-(3-acetylphenyl)-3-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)urea
N-[4-(2-fluorophenoxy)phenyl]-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-2-carboxamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-phenoxyfuran-2-carboxamide
N-(1-ethyl-1H-indazol-3-yl)-2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
(4aR,8aR)-7-(1,3-benzoxazol-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(2-methyl-1-benzothiophen-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-1-[6-(methoxymethyl)pyrimidin-4-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
7-(1,3-benzothiazol-2-yl)-4-[(4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1,9-dimethyl-4-[(2-phenylpyrimidin-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
9-(2-hydroxyethyl)-1-methyl-4-(3,3,3-trifluoropropanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-(morpholin-4-yl)-3-[5-(oxolan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
N-ethyl-5-phenoxy-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]furan-2-carboxamide
methyl 3-(3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamido)propanoate
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
N-[2-(2,4-difluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
4-[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole-5-carbonyl]morpholine
5-(4-benzylpiperidine-1-carbonyl)-1-(cyclohexylmethyl)piperidin-2-one
2-[(dimethylamino)methyl]-4-(1-{[1-(hydroxymethyl)cyclopentyl]methyl}-1H-imidazol-2-yl)phenol
[(2S,4R,5R)-4-{[({3-[2-(dimethylamino)ethoxy]phenyl}methyl)amino]methyl}-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
2-methyl-6-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-4-ol
4-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-tert-butyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
(3S,4R)-N,N-dimethyl-1-(2-phenylquinazolin-4-yl)-4-(propan-2-yl)pyrrolidin-3-amine
7-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-ethyl-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidin-2-one
3-[(dimethylamino)methyl]-1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-ol
1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-ethyl-2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
methyl 3-benzamido-5-{[(2,5-dimethoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-{3-[(pyridin-3-yl)amino]propyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
N,2,6-trimethyl-N-[2-(pyridin-2-yl)ethyl]quinoline-3-carboxamide
{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amine
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
4-[2-(methylsulfanyl)pyrimidin-4-yl]phenol
5-tert-butyl-4-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}furan-2-carboxamide
4-(5-{1-[(2,6-dimethylpyridin-4-yl)methyl]-1H-imidazol-2-yl}pyrimidin-2-yl)morpholine
5-[(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-N,N-dimethylpyridin-2-amine
1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
methyl 5-{[(2-chloro-6-fluorophenyl)methyl]amino}-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]pyridine-3-carboxamide
2-ethyl-5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
3-[(oxolan-2-ylmethyl)sulfamoyl]-N-(pyrimidin-4-ylmethyl)benzamide