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3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-2,8-diazaspiro[4.5]decane
(3-cyclopentylpropyl)(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-{4-[(5-methylthiophen-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
methyl 4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butanoate
N-[(4-fluorophenyl)methyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
2-methyl-1-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}piperidine
N-[(2-fluorophenyl)methyl]-3-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]propanamide
1-(4-{[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}piperidin-1-yl)ethan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
propan-2-yl 4-chloro-3-(pyrrolidine-3-amido)benzoate
1-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(2-phenylpropyl)-1H-1,2,3-triazole
(1S,5R)-3-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(3-methoxyphenyl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)azetidine-1-carboxamide
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]pyridine-3-carbonitrile
(1R,7S)-6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-3-(2-ethylbutyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
4-(2,2-dimethyloxan-4-yl)-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole
2-ethyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)butanamide
(3S,4S)-1-[3-(dimethylamino)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
(2E)-N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-3-(thiophen-2-yl)prop-2-enamide
N-(4-methyl-1,3-thiazol-2-yl)-4-(1-methyl-1H-pyrazol-4-yl)benzamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
3-[2-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
N-[(2-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
1-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
(1R,5S,8R)-8-(dimethylamino)-N-(6-phenoxypyridin-3-yl)-3-azabicyclo[3.2.1]octane-3-carboxamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-(5-methylpyridin-3-yl)urea
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(2,2,2-trifluoroethyl)piperazine
3-[2-(3,4-dimethylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
5-amino-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
1-[benzyl(methyl)amino]-3-{4-[(cyclopropylamino)methyl]phenoxy}propan-2-ol
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
7-[(3-methoxyphenyl)methyl]-2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
5-(2,4-dimethylphenoxy)-1-azabicyclo[3.2.1]octane
6-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-benzyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-thiazole-4-carboxamide
1-(dimethylsulfamoyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-{4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]benzoyl}morpholine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide