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2-[1-(3-phenylpropyl)-4-(1-propylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
2-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
6-(4-methyl-1,4-diazepan-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(1H-indol-5-ylmethyl)acetamide
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-3,5-dimethyl-1H-indole-2-carboxamide
N-cyclopropyl-1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxamide
6-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]pyridine-3-carboxylic acid
2-(benzyloxy)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(pyridin-3-yloxy)acetamide
4-{4-[(3-ethoxy-2-hydroxyphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2-phenylethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
4-(cyclopropylmethyl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
4-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-6-(propan-2-yl)pyrimidin-2-amine
4-(1-propyl-1H-pyrazole-5-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)quinoline
N-[(2,3-dimethylphenyl)methyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
3,6-dimethyl-N-(1,4-oxazepan-6-ylmethyl)-1-benzofuran-2-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
3-ethyl-4-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine-2-carboxylic acid
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
methyl 6-{[bis(prop-2-en-1-yl)amino]methyl}-3-(2-methoxy-2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-methyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-amine
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)propanamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-N-(2-methoxyphenyl)piperidine-1-carboxamide
5-(azocane-1-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
N-methyl-5-{[methyl({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrimidin-2-amine
8-fluoro-2-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}quinoline
1-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
4-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-1-(prop-2-en-1-yl)-1H-pyrazole
N-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]methanesulfonamide
6-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-phenoxy-N-[4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
5-tert-butyl-4-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}furan-2-carboxamide
1-ethyl-3,5-dimethyl-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazole
2-amino-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-{4-[(2-methylpiperidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine
N-methyl-2-{3-[({1-[(3-methylphenyl)methyl]cyclopropyl}carbamoyl)amino]phenyl}acetamide
2-[methyl(pyridin-3-ylmethyl)amino]-1-(1,2-oxazinan-2-yl)ethan-1-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrazolo[1,5-a]pyridine-3-carboxamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(1H-indol-3-yl)ethan-1-one
4-ethyl-5-methyl-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}thiophene-3-carboxamide
2-[3-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetamide