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(1R,5R)-6-(cyclopropylmethyl)-3-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-chloro-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1H-pyrrole-2-carboxamide
N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
7-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroisoquinolin-1-one
1-(2-methoxyacetyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}piperidine-3-carboxamide
1-(morpholine-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{1-[6-(cyclopentylamino)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-{1-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
ethyl 4-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N-cyclopropyl-4-{[3-(pyridin-4-yl)propyl]sulfamoyl}benzamide
N-butyl-2-[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-carboxybutanoyl)pyrrolidine-3-carboxylic acid
3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
2-(2-methoxyphenyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[(3-methoxyphenyl)amino]-N-(2,2,6,6-tetramethylpiperidin-4-yl)butanamide
7-(cyclobutylmethyl)-2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 9-hydroxy-7-oxo-3-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}acetamide
N2,N2,6-trimethyl-N4-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-2,4-diamine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(3-methylthiophen-2-yl)methyl]piperidine
3-[(2R,3R,6R)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,6-difluorobenzamide
6-(piperidin-1-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-4-amine
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-[1-(naphthalen-2-yl)ethyl]propanamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-7-fluoro-3-methyl-1H-indole-2-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
2-methyl-4-(4-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
3-(2-ethylphenyl)-5-methoxypyridine
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[5-(morpholin-4-yl)pentyl]acetamide
N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}-2H-1,3-benzodioxole-5-carboxamide
5-benzyl-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
2-(2,3-difluorophenyl)-1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
3-methyl-4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N,1-dimethyl-4-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-dihydroquinoline-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-{[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
5-{1-[3-(piperidin-1-yl)propanoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(2R,3R)-3-[(2-methoxyethyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-methyl-8-(5-methylthiophene-2-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
methyl(naphthalen-1-ylmethyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide