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2-[(dimethylamino)methyl]-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]benzamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-5-methylphenol
5-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]quinoxaline
methyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(1H-pyrazol-3-ylmethyl)amine
4-{3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
4-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-N-methylbenzene-1-sulfonamide
1-[2-(isoquinolin-1-yloxy)hex-5-en-1-yl]piperidine-4-carboxylic acid
(3S,4R)-4-(3-fluorophenyl)-1-[2-(2-oxoazepan-1-yl)acetyl]pyrrolidine-3-carboxylic acid
5-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
8-(3-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(2-methylfuran-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-{imidazo[1,2-b]pyridazin-6-yl}-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperazine
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2,5-dimethyl-3-(4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)pyrazine
3-[1-(3-hydroxypropyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-methylpropanamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 2-[1-({2-chloro-5-[(propan-2-yl)carbamoyl]phenyl}carbamoyl)pyrrolidin-3-yl]acetate
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(2-methylpropyl)-1H-pyrrole-2-carboxamide
9-(3-methoxybenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2,6-diamino-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]hexan-1-one
N-{3-[4-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}ethane-1-sulfonamide
1-(3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
3-benzyl-4-[3-(furan-2-yl)benzoyl]piperazin-2-one
6-tert-butyl-1-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylbenzoyl)piperidine
3-(2,3-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-[4-(2,3-dimethoxyphenyl)benzoyl]-1H-imidazole
1-{[2-(difluoromethoxy)phenyl]methyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-(1-{imidazo[1,2-a]pyridin-2-ylmethyl}-1H-imidazol-2-yl)-2-(pyrrolidin-1-yl)-1,3-thiazole
4-{[(3-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-methoxy-1-{1'-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]but-3-enamide
[3-(3-methoxypropyl)-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl]methanol
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
3-[(3R,4S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
2-(3-methoxypropyl)-8-(quinolin-5-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-pyrazol-5-yl)benzamide
2-{3-[6-amino-5-cyano-4-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-1H-indol-1-yl}propanoic acid
N-(4-fluorophenyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperazine-2-carboxamide
3-[(2-chlorophenyl)methyl]-N-(1-phenylcyclopropyl)-1,2-oxazole-5-carboxamide
4-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1H-pyrrole-2-carbonitrile