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(1R,9S)-11-{2-methylthieno[3,2-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperidine-4-carboxamide
N4-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
9-(cyclopropylmethyl)-4-methanesulfonyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(diphenylmethyl)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-methyl-8-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-3-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1,2-dihydroquinolin-2-one
5-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
3-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)pyridin-2-amine
1-benzyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-2-({5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)acetamide
6-(2-methoxyphenyl)-N-{1-oxaspiro[4.4]nonan-3-yl}pyridazin-3-amine
5-fluoro-4-(morpholin-4-yl)-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
(E)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-phenylethene-1-sulfonamide
(3S,4S)-4-(dimethylamino)-1-[(2-methylnaphthalen-1-yl)methyl]pyrrolidin-3-ol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(1H-indol-3-yl)acetamide
4-(5-oxo-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepane-1-carbonyl)pyridin-1-ium-1-olate
2-(1-ethenyl-1H-pyrazol-4-yl)-4-(4-ethoxyphenyl)-1H-imidazole
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(2,3,6-trifluorophenyl)acetamide
3-chloro-4-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]pyridine
(1S,5R)-6-(1-methyl-1H-imidazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propylsulfanyl)ethan-1-one
(2S)-2-{[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}-3-(4-hydroxyphenyl)propanamide
(1S,5R)-6-(2-ethoxypyridine-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-4-(1H-imidazol-2-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-ethyl-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-oxazole-5-carboxamide
ethyl 4-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)piperidine-1-carboxylate
8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-5-propyl-1,2-oxazole-3-carboxamide
1-cyclohexyl-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepane
(3R,4R)-1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
4-(1-{4-phenyl-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}ethyl)pyrimidine
1-cycloheptyl-1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
4-[(dipropylamino)methyl]-N-[2-(morpholin-4-yl)ethyl]benzamide
methyl[(1-phenylpyrrolidin-3-yl)methyl](thiophen-2-ylmethyl)amine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
(4aR,7aS)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)methylamine
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
(2R,3S,6R)-3-(3-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(4S)-3,3,4-trimethyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-4-ol
8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclopentyl-N-methyl-5-oxopyrrolidine-3-carboxamide
N,N-diethyl-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
7-chloro-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-methoxy-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol