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4-(3-hydroxy-3-methylbutyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}benzamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-indol-1-yl)ethyl]amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1'-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylthiophene-2-carboxamide
4-{[3-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylaniline
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-methylpiperidin-4-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-(4-methoxyphenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-oxobutanamide
5-ethyl-4-{1-oxa-7-azaspiro[3.5]nonan-7-yl}pyrimidin-2-amine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
(4aS,8aR)-6-cyclopentanecarbonyl-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
[(3,5-dimethoxyphenyl)methyl]({[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl})amine
5-(2-fluorophenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
ethyl 2-{1-[5-(3-acetylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}acetate
2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}pyrazine
3-(cyclopentylsulfamoyl)-5-[3-(hydroxymethyl)phenyl]benzoic acid
N-{2-methyl-1-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}methanesulfonamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(1H-pyrazol-1-yl)benzamide
N-methyl-3-{methyl[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}propanamide
N-(2-methoxyethyl)-1-[1-(pyridazine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-{1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-butyl-N-ethyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(3S,4S)-1-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
5-[4-(benzyloxy)piperidine-1-carbonyl]-2-cyclopropyl-3,4-dihydropyrimidin-4-one
N-(3,5-dimethylphenyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carboxamide
1-(3-methoxyphenoxy)-3-{[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]amino}propan-2-ol
8-(prop-2-ene-1-sulfonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-[methyl(piperidin-4-yl)amino]-N-[1-(2-propoxyphenyl)ethyl]acetamide
5-methoxy-3-methyl-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
4-[3-(3-fluorophenyl)-2-oxo-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]-N,N-dimethyl-4-oxobutanamide
(2S)-N-(1-butyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-phenylpyridazine
8-(2,3-dihydro-1-benzofuran-7-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[4-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
(3S,4S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(pyrrolidine-1-carbonyl)piperidine
ethyl 4-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)piperidine-1-carboxylate
3-{[ethyl(oxan-2-ylmethyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
N3-[3-(4-chlorophenoxy)propyl]-N3-methylpiperidine-1,3-dicarboxamide
N,N-dimethyl-3-[(2-oxoazonan-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide