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1-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-(4-fluorophenyl)-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)acetamide
2-[3-(2-methylpropyl)-5-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl]pyridine
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-ol
N-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
N-(2-methoxyethyl)-3-{1-[4-(4-methoxyphenyl)butan-2-yl]piperidin-4-yl}propanamide
1-methyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
3-{5-[2-(azepan-1-yl)-2-oxoethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
1-(2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
2-(propan-2-yl)-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(5-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}furan-2-yl)methanol
N1,N1-dimethyl-N4-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1,4-dicarboxamide
6-(4-methoxyphenyl)-9-[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanoyl]-6,9-diazaspiro[4.5]decan-7-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
N-[(2R,3R)-2-(benzyloxy)-1'-(furan-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[(2,4-dichlorophenyl)methyl]-2-(trifluoromethyl)morpholine-4-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(9H-purin-6-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
N-[4-(1H-pyrazol-1-yl)phenyl]-6-(1,3-thiazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{3,5-dimethyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
N,1-dimethyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1H-pyrrole-2-carboxamide
1-(furan-2-ylmethyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}piperidine-4-carboxamide
1,3-dimethyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1S,5R)-6-methyl-3-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
2-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-phenylcycloprop-2-ene-1-carboxamide
N-cyclopropyl-2-(dimethylamino)-4-methyl-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-({3-methyl-7-[2-(4-methylphenoxy)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
4-(2-methylphenoxy)-1-[3-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
N-cyclopropyl-3-[5-(1H-indazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclohexyl-N,5-dimethyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1,3-benzothiazol-2-yl)pyrrolidin-3-yl]methanol
(2S,4R)-N-methyl-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-[(pyrimidin-2-yl)amino]pyrrolidine-2-carboxamide
2-{1-[2-(4-fluorophenoxy)ethanesulfonyl]pyrrolidin-2-yl}pyridine
N-[(2R,3R)-1'-[(3,5-dimethylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{1-[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]pyrrolidin-3-yl}acetamide
N-(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-(3-methyl-1H-indole-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,4R)-N-methyl-4-[3-(pyridin-3-yl)propanamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
methyl 4-{[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})carbamoyl}butanoate
1-({1-[(3-ethenylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-ethylurea
(3R,4R)-4-(azepan-1-yl)-1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-ol