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N-{4-[4-(4-cyanophenyl)-2-methyl-5-oxopiperazin-1-yl]-4-oxobutyl}acetamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyridin-4-yl)piperidine-4-carboxylic acid
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
8-methoxy-3-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3,4-dihydroquinazolin-4-one
3-[(3R,4S)-1-[methyl(phenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-chloro-2-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)pyrimidine
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
2,5-dimethyl-N-[4-(pyrrolidin-1-yl)butyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
2-[(4-chlorophenyl)methyl]-N-ethyl-1,3-benzoxazole-5-carboxamide
(8aS)-2-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(6-fluoro-1H-1,3-benzodiazol-2-yl)pyridine-3-carbonitrile
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
3-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-1-ium-1-olate
1-(cyclopropylmethyl)-5-[4-(2-oxopyrrolidin-1-yl)benzoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-oxaspiro[4.5]decan-3-yl}-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
1-(azepan-1-yl)-3-{4-chloro-2-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
3-(3-fluorophenyl)-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
4-[(4-fluorophenyl)methyl]-11-[(2-methoxyethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(9H-fluoren-9-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-(1H-indol-4-ylmethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N,N-dimethylaniline
2-(methoxymethyl)-6-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]pyridine
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-[1-(7-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[2-(2-methylphenyl)ethyl]piperazine
7-(4-chlorophenyl)-2-(pyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2E)-1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-3-(thiophen-2-yl)prop-2-en-1-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(pyridin-3-ylmethyl)acetamide
1-{2-[({3-[2-(methylcarbamoyl)ethyl]phenyl}carbamoyl)amino]ethyl}piperidine-3-carboxamide
5-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione
N-[2-(dimethylsulfamoyl)ethyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-(5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
2-(2,3-dimethoxy-5-methylphenyl)-2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}acetic acid
4-{[1-(furan-2-ylmethyl)piperidin-4-yl]amino}-1-(2-phenylethyl)pyrrolidin-2-one
1-[(1R)-1-(3-methoxyphenyl)ethyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
5-(3,4-dimethoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
4-{[(thiolan-3-yl)amino]methyl}hepta-1,6-dien-4-ol
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-(furan-2-ylmethyl)piperidine
2-{4-[(2-ethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-methyl-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
N-[2-(1H-indol-1-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-[(4aR,7aS)-4-[(4-methyl-1,3-thiazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(1,4-dioxan-2-ylmethyl)(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-[2-(1H-imidazol-4-yl)ethyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine