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7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(cyclohex-3-ene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-6-(6-methoxypyridin-3-yl)-4-(4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-1-methyl-1,2-dihydropyridin-2-one
(4-{4-[(dimethylamino)methyl]phenoxy}phenyl)methanamine
2-{2-[1-(6-cyanopyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-[2-(methylsulfanyl)benzoyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-methoxyphenyl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
2-{4-[4-(diethylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxylic acid
2-(2-phenyl-1H-imidazol-1-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[3-(2-aminoethyl)phenyl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[2-(methylsulfanyl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-3-methyl-1-[4-(methylamino)pyrimidin-2-yl]-4-(oxan-4-yl)piperidin-4-ol
3-methyl-6-[5-(1-phenoxyethyl)-1,2,4-oxadiazol-3-yl]pyridazine
methyl (2S)-2-({2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)-3-methylbutanoate
3,6-dimethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-methyl-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
1-[7-(5-methylthiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
(1S,5R)-3-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(2-hydroxyethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-(4-cyclohexylpiperazine-1-carbonyl)-2-(3-methylphenyl)pyrimidin-4-ol
N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
5-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-fluoro-5-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
(3aR,6aR)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2-methoxyacetyl)-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl N-{[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamoyl]methyl}carbamate
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
7-(3,4-dihydronaphthalen-2-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-ethylpiperazin-1-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(4-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
7-propyl-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(2-aminoethyl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
cyclopentyl 4-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]amino}benzoate
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N1-(6-chloroquinolin-2-yl)ethane-1,2-diamine
1-[(2,6-dimethoxyphenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
(3R,4R)-1-[(3-chlorophenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-[1-(furan-2-ylmethyl)-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
2-[({5-[3-methyl-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)sulfanyl]pyrimidine
4-(3-hydroxybenzoyl)-1-methylpiperazine-2-carboxylic acid
4-{1-[4-(furan-2-yl)butan-2-yl]-1H-imidazol-2-yl}pyridine
2-(methylsulfanyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
4-fluoro-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-(2-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide