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3-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)piperidin-3-ol
ethyl 4-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
4-benzyl-3-ethyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepan-5-one
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,5,6-trimethyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
2-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
5-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-2-(pyridin-2-yl)pyrimidine
N,3,4,7-tetramethyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
N-(4-methoxy-2-methylphenyl)-3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
N-[2-(3-methoxyphenyl)-1-[1-(4-methylpentanoyl)piperidin-4-yl]ethyl]-N,3-dimethylbutanamide
4-(4-chlorophenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-[(4-hydroxyquinazolin-2-yl)sulfanyl]acetamide
N-(2,3-dimethylphenyl)-N'-[(4-fluorophenyl)methyl]-N'-(prop-2-yn-1-yl)propanediamide
N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(4-hydroxyphenyl)benzamide
4-benzyl-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-methoxyphenyl)propanamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(5-methylthiophen-2-yl)methyl]amine
3-methoxy-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}pyridine-2-carboxamide
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
7-acetamido-1-[2-(pyridin-2-yl)ethyl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-[3-(methoxymethyl)pyrrolidin-1-yl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
5-ethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1,3,4-oxadiazol-2-amine
1-benzyl-6-(cyclopropylmethoxy)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-[4-(2-ethyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(4-methoxyphenoxy)ethan-1-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1'-(5-chlorothiophene-2-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N,N-dimethylazepan-4-amine
2-{[cyclopentyl(prop-2-en-1-yl)amino]methyl}pyridine-3-carboxylic acid
5-[2-(morpholin-4-ylmethyl)phenyl]-2-(pyridin-3-yl)-1,3-benzoxazole
2-(2-ethoxy-3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
6-ethoxy-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-[(pyrimidin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
1-methyl-5-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
2-[4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenoxy]pyrimidine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
2-methyl-5-({3-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}sulfanyl)-1,3,4-thiadiazole
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
2-ethyl-9-[(4-methyl-1H-imidazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(2,2-dimethyloxan-4-yl)-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
5-[1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(1S,5R)-6-(2,3-dimethyl-1H-indole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(3S,4S)-1-(2,2-diphenylethyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol