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2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2S)-oxolan-2-ylmethyl]acetamide
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)cyclobutanecarboxamide
N-{2-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
6-(9-methyl-9H-carbazole-3-carbonyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
4-benzyl-3-ethyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1,4-diazepan-5-one
4-(2,4-dimethylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
4-propyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,4-diazepan-5-one
2-amino-3-ethyl-N-[2-(methylsulfamoyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-4-oxo-4-phenylbutanamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}propanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-methylpyridine-3-carboxamide
3-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-(2-fluorophenyl)urea
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
2-(3-hydroxypropyl)-9-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(6-methyl-2H-1,3-benzodioxol-5-yl)pyridine-3-carbonitrile
1-(cyclopropylmethyl)-5-[(4-methylpiperidin-1-yl)sulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methoxyphenyl)methyl]piperidine
3-{5-[2-(morpholin-4-yl)ethyl]-1,3,4-thiadiazol-2-yl}-1-(1,2-oxazol-3-ylmethyl)urea
5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-[3-(dimethylamino)propyl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
4-methyl-3-[(5-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}furan-2-yl)sulfanyl]-4H-1,2,4-triazole
2-(hydroxymethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-1-carboxamide
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide
N-(oxolan-2-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
1-[(2,5-dimethyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)methyl]-2-methylpiperidine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]acetamide
3-(3,4-dichlorophenyl)-1-ethyl-1-(oxan-2-ylmethyl)urea
N-methyl-5-phenyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
2-{4-[(6-methoxy-2H-chromen-3-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-(oxolan-3-yl)-1H-1,2,3-triazole
5-chloro-2-methoxy-4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
1-({5-[1-(2-ethoxyethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
4-[7-(furan-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
5-propyl-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-oxazole
2-({5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)ethan-1-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
3,3-dimethyl-1-{2-oxo-2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}urea
(3aS,6aS)-2-(furan-3-ylmethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-2-{2-[(1-methylpyrrolidin-3-yl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
6-(4-chlorophenyl)-N-[2-(piperidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
[(3R,4S)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(N-methylmethanesulfonamido)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide