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2-[1-cyclopentyl-4-(quinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl 2-[5-methyl-2-({2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]benzoate
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(2-methylpropyl)-1,3-oxazole-4-carboxamide
2-[({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amino]pyridine-4-carbonitrile
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
{1-[3-(azetidine-1-carbonyl)benzenesulfonyl]piperidin-2-yl}methanol
(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)methanol
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylpropanamide
5-(4-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-(4-ethenylphenyl)-2-propylpyrrolidine-1-carboxamide
4-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-2-methylpyrimidine
4-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]quinazoline
(3S)-4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
8-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
2-{[(adamantan-1-yl)amino]methyl}-4-(pyrazin-2-yl)phenol
2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-4-(pyridin-4-yl)pyrimidine
N-cyclopentyl-N'-{[4-(3-fluorophenyl)oxan-4-yl]methyl}butanediamide
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{2-[({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]ethyl}piperidin-4-ol
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-methyl-2-(1H-pyrrol-1-yl)propan-1-one
N-[2-(4-fluorophenyl)ethyl]-2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
1-[1-(4-methylpentyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-methyl-1'-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-propyl-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxylic acid
6-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepane-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-butyl-4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
1-(2-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}phenyl)-1,3-diazinane-2,4-dione
methyl 4-{3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamido}butanoate
4-(ethylamino)-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methylfuran-2-yl)methyl]piperidine-3-carboxamide
4-chloro-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-(2H-1,3-benzodioxol-4-yl)-7-(2-ethoxyethoxy)-1,2,3,4-tetrahydroquinolin-2-one
2-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
6-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
1-[1-methyl-5-(trifluoromethyl)-1H-pyrazole-3-carbonyl]-3-phenylpiperazine
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(naphthalen-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1R,5S)-3-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4,5-dimethylfuran-2-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-(4-methoxyphenyl)-N-[4-(5-methyl-4-{[2-(thiophen-2-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]propanamide
N-[(3S,4R)-1-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-propylpyrrolidin-3-yl]acetamide
1-(4-acetylphenyl)-3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
4-methyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,3-oxazole
1-[(2,4-difluorophenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2S,4S)-4-amino-N-methyl-1-(9-oxo-9,10-dihydroacridine-4-carbonyl)pyrrolidine-2-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(pyrimidin-2-ylsulfanyl)acetamide