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3-(3,4-dimethoxyphenyl)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}propanamide
1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}(4-methoxy-4-methylpentan-2-yl)amine
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-benzyl-3-[1-(but-2-ynoyl)piperidin-4-yl]-N-methylpropanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
N-cyclopropyl-6-(4-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
4-({[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
2-(1-ethyl-1H-pyrazol-4-yl)-N,6-dimethyl-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
2-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
3-({[1-(2,2-dimethylpropyl)cyclopropyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2,4-dichlorophenoxy)-N-(1,4-oxazepan-6-ylmethyl)acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-phenyl-1-[1-(quinoline-3-carbonyl)piperidin-3-yl]ethan-1-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[1-(pyridin-2-yl)propan-2-yl]urea
1-(9H-fluoren-9-yl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
3-{[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
4-benzyl-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(5-methylfuran-2-yl)benzamide
1-[4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N-[(2R,3R)-2-hydroxy-1'-[(3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
5,6-dimethyl-2-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-methyl-N-(2-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}ethyl)pyrazine-2-carboxamide
2-(4-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenoxy)ethan-1-ol
(1R,5R)-6-[(5-fluoro-2-methoxyphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-methyl-N-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
1-[1-ethyl-5-(3-methylthiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
1-[(4-chlorophenyl)methyl]-4-[3-(methylsulfanyl)butyl]piperazine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
2-ethyl-8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4-methyl-6-(trifluoromethyl)pyrimidine
N-({7-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
2-[(1S,5R)-3-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[(3-chlorophenyl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(phenylamino)-N-[2-(pyridin-3-yloxy)propyl]pyrimidine-5-carboxamide
(1r,4r)-4-[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]cyclohexan-1-ol
N-[4-chloro-3-(propylcarbamoyl)phenyl]-4,4-difluoropiperidine-1-carboxamide
3-[(3R,4S)-1-(4-ethenylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2R,3R)-3-[ethyl(methyl)amino]-1'-(5-methylpyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(butan-2-yl)-5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
N,N-dimethyl-N'-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N'-(pyridin-3-ylmethyl)butanediamide
1-[(5-ethylpyridin-2-yl)methyl]-1-methyl-3-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]urea
methyl[(1S)-1-[1-phenyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl]amine