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2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1-[3-(pyrrolidin-1-yl)piperidin-1-yl]ethan-1-one
1-{5-[(2,5-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
6-(4-hydroxyphenyl)-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
5-[(4-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
3-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-phenylbenzamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-(prop-2-en-1-ylsulfanyl)acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-fluoropyridine-4-carboxamide
{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}[(2-methoxyphenyl)methyl]propylamine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]butane-1,2-dione
N-benzyl{[3-(2-methylpyrimidin-4-yl)phenyl]amino}sulfonamide
3-(3,4-dimethoxybenzoyl)-1-(3-fluoro-4-methoxybenzoyl)piperidine
5-{2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
1-({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)-1,4-diazepan-5-one
[(4aS,8aR)-6-propyl-1-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
4-[(4-fluorophenyl)methyl]-1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(4-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]-N-(pyridin-2-ylmethyl)acetamide
8-fluoro-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]quinoline-2-carboxamide
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
1-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-3-(propan-2-yl)urea
1-[(2,6-dimethoxyphenyl)methyl]-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-(1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
7-(1-methylpiperidine-3-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[(4-fluorophenyl)methyl]-5-[1-(4-methylpentanoyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
(2S)-1-{5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propan-2-ol
N-{1-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
{2-[1-(1H-indol-5-ylmethyl)piperidin-2-yl]ethyl}dimethylamine
1-(oxolan-2-ylmethyl)-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
1-(2-methoxyethyl)-8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-methoxy-1H-indol-2-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-cyclopropyl-1-{[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,3-benzodiazole
5-{3-[4-(4-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-methoxy-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-(propan-2-yl)propanamide
2-[(1,3-benzothiazol-2-yl)amino]-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-{[8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
(4aR,8aS)-6-[(4-ethoxyphenyl)methyl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-methyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,3-thiazole-4-carboxamide
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
1-{4-[5-(3-methoxyphenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,4-triazole-5-carboxamide
N-(1-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide