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(2S,4R)-4-amino-N-ethyl-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidine-2-carboxamide
[4-methyl-5-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
2,6-dimethyl-3-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]quinoline
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
{[(1R,5S,6S)-3-[(3,5-dichloropyridin-4-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)azetidin-3-ol
1-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-3-(3-methoxyphenoxy)propan-2-ol
7-(cyclopropylmethyl)-2-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylfuran-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
4-benzyl-3-ethyl-1-[2-(1H-imidazol-1-yl)acetyl]-1,4-diazepan-5-one
3-(3-methoxyphenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-5-carboxamide
7-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
6-chloro-2-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
3-[3-(3,5-dimethylphenyl)propanoyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(1-methyl-1H-indol-3-yl)methyl](pyridin-4-ylmethyl)amine
2,5-dimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
(3aR,5S,6S,7aS)-2-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-octahydro-1H-isoindole-5,6-diol
(1R,2R,4R)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N-[(2,3-dimethoxyphenyl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-N-(thian-4-yl)-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-methyl-N'-(2-methylphenyl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanediamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)amine
2-(adamantan-1-yl)-5-[2-(2-hydroxyethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
(1S,5R)-6-benzyl-3-[2-(3-fluorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(diphenylmethyl)piperazin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
6-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-phenyl-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-2-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
1-(benzyloxy)-8-[3-(prop-2-en-1-yloxy)benzoyl]-1,8-diazaspiro[4.5]decan-2-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyridin-2-amine
methyl 6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-methoxyphenyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-amino-2-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-(1H-indazol-1-yl)ethan-1-one
3-acetamido-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)propanamide
1-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1,3-dimethyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-8-azabicyclo[3.2.1]octane
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(2-methylphenyl)piperidine