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8-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
methyl 3-{[3-(1H-indol-3-yl)propanamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-methyl-N-(oxolan-3-yl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
7-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-ethylbenzamide
2-(1H-imidazol-2-yl)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}benzamide
4-{2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]pyridine-4-carbonyl}morpholine
8-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(4aR,8aR)-7-(1H-1,3-benzodiazol-2-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
2-{[(5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
[(2-fluoro-4-methoxyphenyl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-({8-methyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-[(3S,4R)-4-propyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]methanesulfonamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)cyclopropanesulfonamide
4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
4-(2-methoxybutanoyl)-1-(2-phenylphenyl)piperazin-2-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2,8-dimethylquinoline-3-carboxamide
4-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-amine
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-(2,3-dimethyl-1H-indole-5-amido)pyrrolidine-2-carboxylate
(3S,4R)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-4-(pyridin-2-yl)phenol
1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-({[(4-phenylphenyl)methyl]amino}methyl)phenyl}acetamide
8-[2-(diethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(2-methoxypyridine-4-carbonyl)-1-phenylpiperazin-2-one
2-[4-(1-benzylpiperidin-4-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzenesulfonamide
2-methyl-5-({3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
N-{[1-(3-phenylpropanoyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N,N-dimethyl-5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)furan-2-carboxamide
methyl (2S)-3-methyl-2-[(5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]butanoate
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
6-({4-[1-(cyclohexylmethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-ethyl-5-methyl-6-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
9-(2-hydroxy-3-methoxybenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-phenylethyl)-1-(piperidin-4-yl)piperidine-3-carboxamide
3-[5-(2-methyl-4-phenylpyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-amine
5-(2-phenylazetidine-1-carbonyl)-2-[(phenylsulfanyl)methyl]pyrimidin-4-ol
{3-[(3-chlorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-3-yl}methanol
(5-{4-phenyl-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazol-5-yl}furan-2-yl)methanol
N-[(3-fluorophenyl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide