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1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-amine
4-{4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
5,5-dimethyl-3-{2-oxo-2-[3-(pyrimidin-4-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
(3R)-1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}pyrrolidin-3-ol
4-(2,5-dimethoxybenzoyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N4-[(3,4-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
(5R)-5-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)acetamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(morpholin-4-yl)propan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-N-[2-(2,3-dimethoxyphenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-ethoxy-6-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-({1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}methyl)pyrrolidin-2-one
ethyl 4-{2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamido}piperidine-1-carboxylate
3-({[3-(dimethylamino)propyl](methyl)amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
[3-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenyl]methanol
3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-4-(2-phenylethyl)piperazin-2-one
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
(2-methylpropyl)(pyridin-2-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
N-(1-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
7-(2-methoxyethyl)-2-(6-phenylpyridazin-3-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-phenoxy-N-(1-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
N-[2-(4-fluorophenyl)-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)ethyl]-2-methoxy-N-methylacetamide
9-(cyclopropylmethyl)-1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2,4-dichloro-3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)phenol
1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
(2R)-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxolane-2-carboxamide
2-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
7-propyl-2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-(5-chloropyridine-2-carbonyl)-9-methyl-3,9-diazaspiro[5.6]dodecane
(1R,5S,8R)-N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carboxamide
3-(2-methoxyphenoxy)-1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}azetidine
2-(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}phenoxy)ethan-1-ol
3-{[3-(ethoxymethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
1-ethyl-4-{[methyl({4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl})amino]methyl}pyrrolidin-2-one
N-(2-phenoxyethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-benzyl-3-ethyl-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-5-one