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N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-N,N-diethylpiperidine-3-carboxamide
N-(4-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)acetamide
2-ethyl-N-[(2-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-phenyl-5-(thiophen-3-yl)-1H-imidazole
ethyl 2-chloro-5-{[3-(1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]amino}benzoate
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}butan-1-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
(3R,4R)-3-methyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(oxan-4-yl)piperidin-4-ol
2-[2-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
N-{1-[(4-fluorophenyl)methyl]-7-[2-(2-methoxyethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
N-cyclopropyl-2-{[(3-methylphenyl)methyl]amino}-1-propyl-1H-1,3-benzodiazole-5-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[3-(pyridin-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N-diethyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3,5-dichloro-4-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
6-(2-fluorophenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-chloro-4,6-dimethyl-2-[4-(oxan-4-yl)piperazin-1-yl]pyridine-3-carbonitrile
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}ethan-1-one
2,3,6-trimethyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]quinoline
methyl 7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-(2-hydroxybutyl)-1-(2-methoxyphenyl)piperazin-2-one
3-(5-chloro-2-methoxypyridin-4-yl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(cyclopropylmethyl)-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-propyl-1H-1,3-benzodiazole-7-carboxamide
1-cyclohexyl-4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
N-{2-[4-(dimethylamino)phenyl]ethyl}-3-(1-methylpiperidin-3-yl)propanamide
2-(dimethylamino)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2-fluorophenyl)-N-methylacetamide
N,N-dimethyl-2-[(1S,5R)-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
ethyl 4-{1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carbonyl}piperazine-1-carboxylate
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(2-hydroxypropan-2-yl)pyridine-3-carbonitrile
1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-({2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}(methyl)amino)-N,N-dimethylacetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-propylpyrimidine-5-carboxamide
5-phenyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
4-cyclopentyl-N-[2-(1H-imidazol-1-yl)ethyl]pyrimidin-2-amine
N-[3-(3-methyl-3-phenylpiperidin-1-yl)-3-oxopropyl]methanesulfonamide
{2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}urea
(2S)-2,4-diamino-N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)butanamide
3-(2-phenylethyl)-N-[(4-phenyloxan-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-cyclopropyl-8-(5-fluoro-2-methylbenzenesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-chloropyridine-3-carbonyl)pyrrolidin-3-yl]methanol
1-cyclopentyl-4-{[methyl(quinolin-4-ylmethyl)amino]methyl}pyrrolidin-2-one
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-(furan-3-ylmethyl)piperidine
(2S,4S,5R)-2-ethyl-4-[ethyl(2-hydroxyethyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(furan-2-carbonyl)piperidin-4-yl]propanamide
7-fluoro-3-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1-benzofuran-2-carboxamide
6-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]quinoline
3-[({[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]piperidin-3-ol
2-methyl-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-2-(thiophen-2-ylformamido)propanamide