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3-cyclopropyl-6-(4-phenylbutyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-ethoxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
8-(3-methoxypropanoyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(pyridin-2-yl)propanoyl]piperidine-3-carboxylate
methyl 5-[(1-benzofuran-2-ylmethyl)amino]-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(4-ethenylbenzoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-(2-fluorophenyl)acetamide
1-(4-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
3-(5-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-(3-chloro-4-methoxyphenyl)-3-cyclopropyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(9H-fluoren-9-yl)propanamide
1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(3S,4S)-4-(dimethylamino)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
3-{3-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
N,N-dimethyl-6-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-4-amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]urea
2-(4-{1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propanamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1R)-1-(4-methoxyphenyl)ethyl]propanamide
[(2S,6S)-4-(4-methoxypyrimidin-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[(4-methoxyphenyl)methyl]-4-[4-(pyrrolidin-1-yl)pentanoyl]piperazin-2-one
(4aS,8aR)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
1-({1-[6-(3-methylphenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
(2R,6S)-4-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
2-(dimethylamino)-N-ethyl-4-methyl-N-(oxan-4-ylmethyl)pyrimidine-5-carboxamide
1-[(3S,4R)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(2E)-3-(4-methoxyphenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)prop-2-enamide
3-(2-hydroxyphenyl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1H-pyrazole-5-carboxamide
1-(2-chlorophenyl)-2-{4-[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethan-1-ol
N-(2-fluorophenyl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
methyl 7-oxo-3-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(2-fluorophenoxy)-1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
N-methyl-N-[2-(2-methylphenyl)-1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide
9-{2-[methyl(phenyl)amino]acetyl}-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(propan-2-yl)-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
N-ethyl-3-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide
2-(3-methoxyphenyl)-1-(2-methyl-1-benzofuran-5-carbonyl)azetidine
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](furan-2-ylmethyl)methylamine
3,5-dimethyl-N-(3-phenylpropyl)-1-benzofuran-2-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
{2-methoxy-5-[2-(morpholin-4-ylmethyl)phenyl]phenyl}methanol
N-cyclopropyl-1-[1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-(pyrrolidine-1-carbonyl)piperazine
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
N,N-dimethyl-1-{1H,3H,4H,5H-thiopyrano[4,3-b]indole-8-carbonyl}azepan-4-amine
3-({2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazol-5-yl}formamido)-N,N-dimethylpropanamide
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 4-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]piperidine-1-carboxylate
1-(benzyloxy)-8-(2-chloro-6-fluorobenzoyl)-1,8-diazaspiro[4.5]decan-2-one
1-[2-(naphthalen-2-yloxy)propanamido]cyclopentane-1-carboxylic acid