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2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-N-(2-methoxy-5-methylphenyl)acetamide
methyl 4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-4-oxobutanoate
(3S,4S)-N-[4-(2-fluorophenoxy)phenyl]-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
2-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
1-(4-{4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}phenyl)ethan-1-one
1-[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]-1,4-diazepan-5-one
1-methyl-9-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(2S,4R)-4-amino-N-ethyl-1-[4-(5-methylfuran-2-amido)benzoyl]pyrrolidine-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-cyclopropyl-1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
methyl 5-{[1-(dimethylamino)propan-2-yl]amino}-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3-phenylpiperazine
5-ethyl-2,3-dimethyl-N-[5-(morpholin-4-yl)pentyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
12-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
1-(1H-indol-4-ylmethyl)-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[(4-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
1,5-dimethyl-4-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
5-{1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
N-[2-(furan-2-yl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
3-fluoro-N-[(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
3,5-difluoro-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}pyridine
2-(1H-imidazole-2-carbonyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-(1H-1,3-benzodiazol-2-yl)-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
N,N-diethyl-1-[(1s,4s)-4-[2-(1-methyl-1H-pyrrol-3-yl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(but-2-ynoyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]ethan-1-one
1-(4-methyl-2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}pyrimidin-5-yl)ethan-1-one
3-(1H-indol-3-yl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]propanamide
5-(4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
4-[5-(naphthalene-2-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-(2-methoxy-4-methylphenoxymethyl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(methoxymethyl)piperidine
1-[(3,4-difluorophenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
2-(1-cyclohexyl-5-{2,7-dimethylimidazo[1,2-a]pyridin-3-yl}-1H-1,2,4-triazol-3-yl)acetamide
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-(piperidin-4-yl)pyridine-3-carbonitrile
1-(2-methylpropyl)-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrrolidin-2-one
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[4-methyl-3-(propan-2-yl)phenyl]-1-[1-(pyrazin-2-yl)propan-2-yl]urea
dimethyl[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)methyl]amine
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}cyclobutanamine
(4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methanol
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
4-{[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]sulfonyl}benzoic acid