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2-[1-(propan-2-yl)piperidin-4-yl]-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[({1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
5-ethyl-4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazole
N-(1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
4-(2-hydroxypyridine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
1-[benzyl(methyl)amino]-3-(5-{[ethyl(2-hydroxyethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-1,3-benzodiazole
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
1-methyl-8-[2-(4-methylphenyl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
5-methoxy-9-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
(2S)-1-acetyl-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
8-(butan-2-yl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,7S,8aS)-7-[(1-benzothiophen-2-ylmethyl)amino]-3-[(4-chlorophenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(1R,3s,6r,8S)-4-{5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
N-[2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-3-carboxamide
N-(2-methoxyethyl)-3-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-cyclohexyl-3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-imidazole-2-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenylethan-1-one
3-{1-[2-(1H-imidazol-4-yl)acetyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
5-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
ethyl 4-[(2-chlorophenyl)methyl]-1-(3-fluorobenzenesulfonyl)piperidine-4-carboxylate
2-{4-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperazin-1-yl}phenol
2,4-dioxo-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
2-{4-[4-(ethylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-indazol-3-yl)acetamide
4-(5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-{2-amino-4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(furan-2-yl)propan-1-one
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-6-methyl-1,2-dihydroquinolin-2-one
2-(5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
2-(4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-methyl-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-thiazole-4-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-methylpyridin-4-yl)methyl]benzamide
N-methyl-5-(oxolan-2-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
3-(4-ethylphenyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
2-(furan-2-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-oxoacetamide
2-methyl-6-[1-(4-methylquinolin-2-yl)piperidin-4-yl]pyrimidin-4-ol
2-(2,7,8-trimethylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
N,N-dimethyl-1-(2-methylpropyl)-5-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide