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1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
5-[1-(2-acetylbenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(4-methoxyphenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentane-1-carboxamide
N-[(2-methoxyphenyl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
[5-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
2-[2-(dimethylamino)ethyl]-9-(2-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)methyl]benzamide
3-[(dimethylamino)methyl]-1-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperidin-3-ol
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
2-{1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-{2-[2-(2-chlorophenyl)-1H-imidazol-1-yl]ethyl}-4-(2-methoxyethyl)-4H-1,2,4-triazole
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(piperidin-3-yl)pyridin-2-amine
5-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methyl-1,4-dihydropyridin-4-one
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-phenoxyethyl)piperazine
(2S,4R)-4-(2H-1,3-benzodioxole-5-amido)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrrolidine-2-carboxamide
2,5-dimethyl-N-{2-[5-methyl-4-({[3-(prop-2-en-1-yloxy)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-3-carboxamide
4-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
2-(2-methoxy-4-methylphenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-(adamantan-1-yl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-[4-(benzylamino)piperidin-1-yl]-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[2-(cyclopropylmethyl)-4-[(1-methylpiperidin-4-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
(2-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}phenyl)methanol
N-(cyclobutylmethyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(oxolan-2-ylmethyl)propanamide
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[2-(3-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophen-2-yl]ethan-1-one
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(2S,4R)-N-ethyl-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-propanamidopyrrolidine-2-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-ol
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(pyridin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-butyl-N-(furan-2-ylmethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
4-[2-(4-fluorophenyl)morpholin-4-yl]-2-methoxypyridine-3-carbonitrile
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
N-[(1-methylpyrrolidin-3-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1,3-benzoxazole
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
N-({7-[2-(2-chloro-4-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
7-(cyclopropylmethyl)-2-(quinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2-methylpropyl)({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-2-ylmethyl)amine
N-cyclooctyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
3-(2-methoxyphenyl)-1-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]propan-1-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-3-carboxylate
1-ethyl-N-(2-hydroxyethyl)-4,6-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1-methyl-1H-pyrazole