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2-{[(3-cyano-2-methoxypyridin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenoxy}pyrimidine
4-({4-methyl-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-{1-[(5-methylpyrazin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
2-cyclopropyl-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
2-(4-methyl-6-{[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}pyrimidin-2-yl)phenol
6-[(2-chloro-4,5-dimethoxyphenyl)methyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
7-methyl-4-oxo-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-4H-chromene-2-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-(3-ethoxypropyl)-6-oxopiperidine-3-carboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[2-(4-methylbenzoyl)-1H-imidazol-1-yl]acetamide
4-(2,6-dimethylpyridin-3-yl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
3-acetyl-N-[3-(2-methoxyphenyl)-3-methylpentyl]-1H-pyrazole-5-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(quinolin-3-ylmethyl)amine
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-3,4-dihydrophthalazine-1-carboxamide
methyl 4-{4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazol-1-yl}butanoate
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-3-amine
2-[2-(1H-imidazol-4-yl)ethyl]-9-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-(cyclopentylamino)-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
methyl 2-(3-{[benzyl(ethyl)amino]methyl}-7-chloro-2-oxo-1,2-dihydroquinolin-1-yl)acetate
6-(4-fluorophenyl)-N-methyl-N-(quinolin-6-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1S,5R)-6-(5-methylpyrazine-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-amine
3-methoxy-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
6-[(2,3-dihydro-1H-inden-2-yl)amino]-2-methylheptan-2-ol
1-{2-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-(3-tert-butyl-1,2,4-oxadiazol-5-yl)quinoline
1-(4-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
2-amino-4-(2-methoxypyrimidin-5-yl)-6-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
7-(3-methoxypropanamido)-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2,5-dimethoxybenzamide
N-(1-ethyl-1H-pyrazol-5-yl)-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
N-[(3-chlorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
N-(2,4-dimethoxyphenyl)-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-{[3-(2-aminoethyl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1'-(dimethyl-1,3-thiazole-5-carbonyl)spiro[indene-1,4'-piperidine]
(2S)-2-[1-(4-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
2-cyclopentyl-N-[3-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
2-(1H-1,3-benzodiazol-1-yl)-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
propyl({[3-(1H-pyrazol-3-yl)phenyl]methyl})amine
6-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
8-[2-(methylsulfanyl)pyrimidin-4-yl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[3-(dimethylamino)-2-hydroxypropyl]piperazin-1-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one