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(4aR,8aR)-2-[(2-fluoro-4-methoxyphenyl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
4-ethyl-1-methyl-3-({1-[4-(pyrrolidin-1-yl)butanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-methyl-9-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
9-[2-(phenylsulfanyl)ethyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
1-ethyl-3-(thiomorpholine-4-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4S)-1-(2,5-dimethylfuran-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
4-[3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
3-[(2-methylphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
N-(2-phenylethyl)-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2-cyclopropyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
N-(3-methyl-1,2-oxazol-5-yl)-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
3-[2-(2,6-difluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[1-(1-benzylpyrrolidine-2-carbonyl)azetidin-3-yl]pyridine
6-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)piperidine-3-carboxamide
4-(1,3-benzothiazol-6-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2E)-N-({7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
(4-{[1-(1-methyl-1H-indole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-benzyl-2-hydroxy-N-(3-hydroxy-2-methylpropyl)-5-methylbenzamide
4-[(4-fluorophenyl)methyl]-1-(5-fluoropyridine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
ethyl 4-[2-(3-fluorophenyl)-1,3-benzoxazole-5-amido]piperidine-1-carboxylate
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
N,4-dimethyl-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}amino)benzamide
3-[5-chloro-2-(propan-2-yloxy)phenyl]-[1,2,4]triazolo[4,3-a]pyridine
3-(2-methoxyethyl)-5-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazole
1-(3-fluoropyridin-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
5-acetyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)(methyl)amino]propanamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[4-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1H-imidazol-1-yl)-1-(2-methylquinolin-4-yl)piperidine-4-carboxylic acid
2-{1-benzyl-5-[(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
(1-{1-[3-(azepane-1-carbonyl)-6-(2-methoxyphenyl)pyridin-2-yl]piperidin-4-yl}piperidin-3-yl)methanol
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-(pyridin-4-yl)piperazine
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
5-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
benzyl({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-(3-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenoxy)ethan-1-ol
1-(2,7-dimethylquinoline-4-carbonyl)-2-methyl-1,4-diazepan-5-one
5-methyl-2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-imidazole-4-carboxamide
2-[(2-chlorophenyl)methyl]-4-(pyrazine-2-carbonyl)morpholine
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(2-phenylethyl)acetamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-N-{[2-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
6-(4-chlorophenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 5-[(furan-2-ylmethyl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate