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{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
4-(1-benzofuran-5-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
6-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{1-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]azetidin-3-yl}piperidine
6-methyl-3-[3-(pyridin-3-yl)azetidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-{2-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)pyrrolidin-3-yl]methyl}prop-2-ene-1-sulfonamide
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-ol
2-(4-methyl-6-{[1-(pyrimidin-4-yl)ethyl]amino}pyrimidin-2-yl)phenol
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
(3S,4R)-4-(hydroxymethyl)-1-[4-(3-methylphenoxy)benzoyl]piperidin-3-ol
4-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperazin-2-one
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[3-(1,3-thiazol-4-yl)phenyl]-1-(thiophen-2-ylmethyl)piperidine-4-carboxamide
1-{3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-(oxan-4-ylmethyl)acetamide
4,6-dimethyl-1-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,2-dihydropyrimidin-2-one
2-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)amino]pyridine-4-carboxamide
4-methyl-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentan-1-one
N-[3-(1H-indol-2-yl)phenyl]-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-3-carboxamide
5-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(cyclopropylmethyl)(oxolan-2-ylmethyl)amine
2-{3-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
3-[(2R,3R,6R)-5-(2,6-difluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-(4-chlorophenoxy)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-4-carboxamide
6-ethyl-2-methoxy-3-[({7-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(2-methoxyethyl)-6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-3-carboxamide
methyl 1-{1-[3-(2-oxopyrrolidin-1-yl)phenyl]piperidin-4-yl}piperidine-4-carboxylate
3-(3-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
3-(1H-indol-5-yl)-5-(morpholine-4-sulfonyl)benzoic acid
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-benzyl-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(2-fluorophenyl)methyl]({[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
(2E)-3-(4-methoxyphenyl)-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
N-{[(3S,4S)-3-hydroxy-1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl]methyl}-3-methylbenzamide
ethyl 1-{3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidine-3-carboxylate
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(4-methoxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-N-methylpiperidine-2-carboxamide
N-{2-[1-(2,5-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-(4-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
N-({7-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-(2-methoxyethyl)-1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-(piperidin-1-ylmethyl)phenoxy]propan-2-ol
4-fluoro-N-[2-({2-oxo-1-oxaspiro[4.5]decan-4-yl}formamido)ethyl]benzamide
(3S,4S)-4-(dimethylamino)-1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}benzamide
N-benzyl-3-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-methylpropanamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-3-carboxamide
N-[(1R,3S)-3-{[2-(methylsulfanyl)phenyl]carbamoyl}cyclopentyl]morpholine-4-carboxamide