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2-(3-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydro-1H-isoindole
2-{4-[(2,5-difluorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
4-methyl-2-phenyl-6-[3-(piperidin-1-yl)azetidin-1-yl]pyrimidine
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]-1,2-oxazole-3-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
4-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
2-(3-hydroxypropyl)-9-[2-(4-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidine-1-carboxamide
1-methyl-8-{[2-(methylsulfanyl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[1-(1-methyl-1H-pyrazol-5-yl)-N-(2-phenylethyl)formamido]propanamide
(1S,5R)-6-propyl-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]amine
2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
8-(ethanesulfonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3,4-difluorophenyl)methyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
({5-[(3-fluoropyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-propoxypiperidine
4-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol
4-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}methyl)benzene-1-sulfonamide
5-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-2-hydroxybenzoic acid
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-[1-(thiophen-2-yl)ethyl]propanamide
3-(2-ethoxypyridine-3-carbonyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
6-phenyl-3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-3-(3-methylphenyl)piperidine
1-(1,3-benzothiazol-6-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(3-methylbutyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2-[1-(pyridin-2-ylmethyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-cyclopropyl-2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
4-benzyl-N-(2,4-dimethoxyphenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methanol
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
1-(benzyloxy)-3-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-2-ol
ethyl 1-{1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carbonyl}piperidine-4-carboxylate
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-N-[(2-chlorophenyl)methyl]propanamide
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-(4-methanesulfonylphenyl)-1-[3-(4-methylpiperazin-1-yl)propyl]urea
6-methyl-N4-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-2,4-diamine
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
3-(azepane-1-carbonyl)-1-ethyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[9-(3-fluoropyridin-4-yl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-(1-ethylpiperidin-4-yl)-5-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine