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5-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(3-methylbutyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(3-methoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(2S)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxolane-2-carboxamide
2-(1H-pyrazol-1-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]-1,4-oxazepane-4-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[1-(4-fluorophenyl)propyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(2,3-dihydro-1H-inden-1-yl)acetamide
methyl 5-(cyclohexylamino)-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(4,4-diphenylpiperidin-1-yl)-2-oxoethyl]-5-methylpyrrolidin-2-one
2-(8-methoxy-2-methylquinolin-5-yl)-1,3-thiazole-4-carboxamide
4-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
5-cyclobutanecarbonyl-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
9-methoxy-7-(5-methylthiophen-2-yl)-4-(2-propoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
N-benzyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-(2-phenylethyl)acetamide
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-hydroxy-2-methylpropan-1-one
1-[(1S,5R)-6-(2,3,4-trimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-({1-[3-(4-chlorophenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
2-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
5-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidin-4-ol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(3-methoxypropyl)piperidine-3,5-dicarboxamide
1-(adamantan-1-yl)-4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperazine
1-butyl-3-[2-(methylsulfanyl)ethyl]-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-(1-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylpyridine-3-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-N,N-dimethylbenzamide
6-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(2,3-dimethoxyphenyl)methyl](2-methoxyethyl)amine
2-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-[1-(1-ethylpiperidin-4-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-[2-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-3-ol
methyl 3-(2-methoxybenzamido)-5-{[2-(4-methoxyphenoxy)acetamido]methyl}benzoate
N-({7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
6-(3-propyl-1H-pyrazole-5-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
1-ethyl-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-cyclopropyl-6,6-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-5-oxothiomorpholine-3-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-1,2,4-triazine
3-{[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-cyclopropyl-5-(2-fluorophenoxymethyl)-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-[2-(pyrrolidin-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
6-[(4-fluorophenyl)methyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-({7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(oxolane-2-carbonyl)piperazine
1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-methoxypropan-1-one