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2-ethoxy-5-[2-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]benzoic acid
1-(furan-2-ylmethyl)-4-(pyrazin-2-yl)-1,4-diazepane-6-carboxylic acid
2-[(3S,4R)-3-cyclopropyl-4-(5-phenylpentanamido)pyrrolidin-1-yl]acetic acid
4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
methyl 8-(1H-indol-3-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
(1R,5R)-6-[(2,5-difluorophenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-(cyclopropylmethyl)-5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclopropyl-N-{2-[methyl(phenyl)amino]ethyl}-5-oxopyrrolidine-3-carboxamide
5-{[(3R,4S)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]methyl}-N-methylfuran-2-carboxamide
1-[2-hydroxy-3-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
2-amino-7-methoxy-4-(pyridin-4-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
3-{[1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}benzamide
5-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[5-(oxolan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
2-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(methylamino)-N-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}benzamide
N-methyl-N-[1-(pyridin-3-yl)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}pyrrolidin-3-yl]methanol
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-3-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}propanamide
methyl 2-[(cyclopropylmethyl)(propyl)sulfamoyl]-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
dimethyl(2-{5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)amine
4-[(4-fluorophenyl)methyl]-N-(1H-indazol-6-yl)-1,4-diazepane-1-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
[2-(2,3-dihydro-1,4-benzodioxin-6-yl)quinolin-3-yl]methanol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-methyl-1,3-benzoxazole-6-carboxamide
4-{[butyl(furan-2-ylmethyl)amino]methyl}-N-methylbenzene-1-sulfonamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-benzyl-5-acetamido-2-methyl-1H-1,3-benzodiazole-7-carboxamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[(4-phenyloxan-4-yl)methyl]piperidin-4-amine
(3aR,6aS)-5-[3-(methylsulfanyl)propyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-2-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)acetamide
1-(3-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1-methyl-1H-1,2,4-triazol-5-yl)piperidine
2-(ethylamino)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyridazine-4-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
(3S,4R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
{4-benzyl-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-4-yl}methanol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(2E)-3-(pyridin-2-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(2-fluorophenyl)pyrrolidine-2,5-dione
3-(3-chloro-1,2-oxazol-5-yl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}propan-1-one
8-cyclopentyl-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-(furan-2-yl)ethyl](methyl){[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amine
(1R,3S)-3-(2-aminoethoxy)-7-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-7-azaspiro[3.5]nonan-1-ol