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2-{2-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
N4-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-2,4-diamine
4-benzyl-2-{2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
(1R,7S)-3-tert-butyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{3-[3-(1H-pyrazol-1-yl)phenyl]phenyl}-4H-1,2,4-triazole
methyl 1-(3,4-dihydro-2H-1-benzopyran-3-yl)piperidine-4-carboxylate
2-(4-{3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazin-1-yl)quinazoline
3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-N-(4-methylpyridin-2-yl)propanamide
N-(1-benzylpiperidin-4-yl)-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(butane-1-sulfonyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
1-(1-benzothiophene-5-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2-{1-[(2-ethoxyphenyl)methyl]-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
8-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-(2-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-yl}ethyl)phenol
N-[2-(oxolan-3-ylformamido)ethyl]pyridine-3-carboxamide
1-[(1-ethyl-2-methyl-1H-1,3-benzodiazol-5-yl)oxy]cyclohexane-1-carboxylic acid
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylacetamide
N-[(5-chlorothiophen-2-yl)methyl]-2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzamide
6-(2-phenoxyphenyl)-1H-[1,2,3]triazolo[4,5-b]pyridine
2-[5-cyclopropyl-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2,5-dimethylthiophen-3-yl)pyrimidine
1-tert-butyl-4-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}pyrrolidin-2-one
methyl 3-{[2-(1H-1,3-benzodiazol-1-yl)acetamido]methyl}-5-(2-chlorobenzamido)benzoate
methyl 4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]benzoate
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
2-fluoro-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
4-(5-{1-[(4,6-dimethylpyrimidin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}-1,3-thiazol-2-yl)morpholine
5-(2,3-dihydro-1,4-benzodioxin-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-(methoxymethyl)-1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]acetate
3-(furan-2-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2,2-dimethyl-N-{2-methyl-3-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]phenyl}propanamide
(2E)-2-methyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-2-enamide
5-tert-butyl-4-[(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)methyl]furan-2-carboxamide
N-butyl-3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methylbenzamide
methyl 4-({[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)benzoate
4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-N-phenylpiperidine-1-carboxamide
1-(1H-pyrrole-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-methyl-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-4H-1,2,4-triazole
9-(4-chloro-1H-indole-2-carbonyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-{2-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]ethyl}acetamide
1-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
methyl 2-[3-(3-chlorophenyl)-N-methyl-3-phenylpropanamido]acetate
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4S)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-cyclooctyl-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)acetamide
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(pyrrolidin-1-yl)pyrimidine
2-(2-oxo-2-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide