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1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazole
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-imidazole-2-carboxamide
2-methyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-1,3-thiazole-4-carboxamide
3-({[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
9-methoxy-3-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[3-benzyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(2S)-1-hydroxypropan-2-yl]acetamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(oxane-4-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(propan-2-yl)-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyridin-3-ol
N-[2-(dimethylamino)ethyl]-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(4-methoxypyrimidin-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N-[(2R,3R)-1'-[3-(furan-2-yl)propanoyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-[3-(dimethylamino)propyl]-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
2-(3-methylbutyl)-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
1-(2-aminoethyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
{3-[(4-fluorophenyl)methyl]-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methanol
N-[1-(2-chlorophenyl)ethyl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(4-fluorophenyl)-N-(2-{7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-{[1-(dimethylamino)cycloheptyl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-cyclohexyl-N-cyclopropyl-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-({[(2-chlorophenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1,3-dimethyl-5-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(1H-imidazol-2-ylmethyl)-4-(4-methoxyphenoxymethyl)piperidine
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
[(3R,4R)-1-(furan-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-({2-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
(3aS,7aR)-5-methyl-2-(4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-fluoro-2-[1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-(2-methoxyphenyl)-2-methyl-1-(4-methyl-1,3-thiazol-2-yl)piperazine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxane-4-carbonyl)piperidine
ethyl 5-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(2-chlorophenyl)methyl]-N-methyl-N-[4-(morpholin-4-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
4-(pyrazin-2-yl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3λ6,4-oxathiazinane-3,3-dione
{1-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidin-3-yl}methanol
1-[(6-methylpyridin-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
ethyl 4-{[2-hydroxy-5-(2-methylquinolin-4-yl)phenyl]methyl}piperazine-1-carboxylate
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[(2S,6S)-4-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-hydroxy-2-phenylethyl)-N-methylpropanamide
2-cyclobutanecarbonyl-6-methyl-5-[5-(4-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine