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N-({1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-3-yl}methyl)furan-2-carboxamide
1-{3-oxo-3-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propyl}pyrrolidin-2-one
2-{5-[3-(morpholin-4-yl)butyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
1-[3-({4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylpropanamide
N-cyclopropyl-2-[4-(2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetyl)morpholin-3-yl]acetamide
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
4-[4-(pyridin-4-yl)pyrimidin-2-yl]morpholine
ethyl 5-({[1-(4-{[(3S)-2-oxoazepan-3-yl]carbamoyl}phenyl)piperidin-4-yl]amino}methyl)furan-2-carboxylate
4-benzyl-3-[1-(2,2-dimethylcyclopropanecarbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{5-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-(2-phenylpropyl)piperidin-4-ol
4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepane-1-carbaldehyde
4-({2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
N-methyl-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)-N-(quinolin-5-ylmethyl)acetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[(2R,3R)-1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
5-(4-methyl-1,4-diazepan-1-yl)-2-(pent-2-yn-1-yl)-2,3-dihydropyridazin-3-one
3-(benzyloxy)-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1,5-dimethyl-1H-indazole
1-(4-carbamoylpyridin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-(1H-indol-2-ylmethyl)-3-methoxybenzamide
N-ethyl-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1,6-dihydropyridine-3-carboxamide
5-chloro-N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2-methoxybenzene-1-sulfonamide
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
N-(1H-indol-2-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethyl}morpholine
2-({[2-(dimethylamino)ethyl](ethyl)amino}methyl)-4-(pyridin-3-yl)phenol
3-methoxy-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propan-1-one
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-(benzylamino)-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
8-(2-cyclopentylacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
(3R,9aR)-8-(cyclopropylmethyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-butyl-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3,4-difluorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-ethyl-N-(oxolan-2-ylmethyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
4-{[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-3-yl]methyl}morpholine
3-methyl-3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-(1H-1,2,3,4-tetrazol-5-yl)urea
N,N,4-trimethyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
7-(5-methoxy-1H-indole-2-carbonyl)-2-oxa-7-azaspiro[4.5]decane
6-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-[4-(1H-pyrazol-1-yl)phenyl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
2-(3,5-dimethoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]acetamide