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3-[(3R,4S)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N,N-dimethyl-2-{[(3-methylthiophen-2-yl)formamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{[2-(3-acetyl-2-fluorophenyl)phenyl]methyl}propanamide
ethyl 1-(cyclopropylmethyl)-5-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[4-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N3-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-N5-[(4-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1-(isoquinolin-5-yl)urea
2-[(3,4-dimethoxyphenyl)methyl]-N-(1H-indol-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
(3-{2-[1-(2-ethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-[4-(4-fluorophenyl)piperazin-1-yl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-methyl-N-(2-phenyl-1-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
(3aS,7aR)-2-[2-(2-methoxyethoxy)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[4-(3-methylphenoxy)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1H-indol-3-yl)ethyl]acetamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3R,6R)-5-cyclopropanecarbonyl-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(3-methylbutyl)-5-{1-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[(2-chlorophenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)morpholine
methyl 3-[4-(4-methoxyphenyl)butan-2-yl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(oxolan-2-ylmethyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
1-cyclohexyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpiperidine-4-carboxamide
2-{[methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]methyl}benzoic acid
4-(4-chlorophenyl)-1-[7-(pyrrolidin-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(5-methylfuran-2-yl)benzamide
3-benzyl-5-(2-methoxyphenoxymethyl)-1H-1,2,4-triazole
6-(1-ethyl-6-oxopiperidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-({7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
5-methyl-N4-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyrimidine-2,4-diamine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
1-[(2-methoxyphenyl)methyl]-N-[(5-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}piperidin-2-one
(4aR,7aS)-1-benzyl-4-[(3-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4S)-1-(5-methylthiophene-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(1-benzothiophen-2-ylmethyl)({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-phenyl-N-{4-[4-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidin-1-yl]phenyl}propanamide
N-{1-[({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
N-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}oxolane-2-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}but-3-enamide
(1R,5S,8S)-3-({3-[3-(dimethylamino)propoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
3-ethyl-1-(quinoline-4-carbonyl)piperidine-3-carboxylic acid
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
5-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}pyrazin-2-ol
(2S)-1-acetyl-N-[(3-chlorophenyl)methyl]-N-propylpyrrolidine-2-carboxamide
1-({5-[(2-methoxy-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea